SCHEMBL3470074

SCHEMBL3470074

Cc1ccc(N(C(=O)OC(C)(C)C)S(=O)(=O)c2cccc(C#CCC(C)(CCc3ccc(-c4cccc(C#N)c4)cc3)C(=O)O)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 3/20 0.43
PTPN2 P17706 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPRS Q13332 1/20 0.43
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
MCHR1 Q99705 6/20 0.37
HRH3 Q9Y5N1 5/20 0.37
PTGER1 P34995 1/20 0.35
ACLY P53396 1/20 0.35
PTGER2 P43116 1/20 0.34
STAT5B P51692 1/20 0.34
ADAMTS4 O75173 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
NR1H3 Q13133 1/20 0.33
NR1H2 P55055 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3469959 0.89 STAT3 (0.42) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL3467263 0.84 PTPN2 (0.39) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL3469957 0.78 PTPN2 (0.40) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL1860642 0.77 CA12 (0.38) STAT5B
SCHEMBL3465873 0.76 MMP13 (0.42) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL3466770 0.74 MMP13 (0.45) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL1855155 0.74 STAT5B (0.37) MMP13STAT5B
SCHEMBL1855996 0.73 STAT5B (0.36) MMP13STAT5B
SCHEMBL3467062 0.73 MMP13 (0.43) STAT3PTPN2PTPN1PTPRSMMP12
SCHEMBL1857094 0.72 F2 (0.40) NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO disclosed