SCHEMBL3465873

SCHEMBL3465873

CC(C)(C)OC(=O)N(c1ccccc1)S(=O)(=O)c1ccc(C#CCC(CCc2ccc(-c3cccc(C#N)c3)cc2)C(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 12/20 0.42
MMP12 P39900 1/20 0.42
MMP2 P08253 11/20 0.40
ADAMTS4 O75173 2/20 0.39
PTPN2 P17706 1/20 0.38
PTPN1 P18031 1/20 0.38
STAT3 P40763 1/20 0.38
PTPRS Q13332 1/20 0.38
MMP3 P08254 9/20 0.37
MMP1 P03956 4/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
FFAR1 O14842 1/20 0.34
CTSB P07858 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PTGER2 P43116 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3466770 0.90 MMP13 (0.45) MMP13MMP12MMP2ADAMTS4PTPN2
SCHEMBL3467062 0.85 MMP13 (0.43) MMP13MMP12MMP2ADAMTS4PTPN2
SCHEMBL3467263 0.83 PTPN2 (0.39) MMP13MMP12ADAMTS4PTPN2PTPN1
SCHEMBL1859570 0.80 MMP13 (0.38) MMP13MMP2MMP3MMP1MMP9
SCHEMBL1861012 0.79 TP53 (0.37) MMP13MMP2MMP3MMP1MMP9
SCHEMBL1861139 0.78 ALDH1A1 (0.36) MMP13MMP2MMP3MMP1MMP9
SCHEMBL3470074 0.76 STAT3 (0.43) MMP13MMP12ADAMTS4PTPN2PTPN1
SCHEMBL3469957 0.76 PTPN2 (0.40) MMP13MMP12ADAMTS4PTPN2PTPN1
SCHEMBL1855155 0.74 STAT5B (0.37) MMP13MMP2MMP3CTSSCTSK
SCHEMBL1856286 0.73 KMT2A (0.40) MMP13MMP12MMP2STAT3MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO claimed
WO-2010070076-A1 ALKANOIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE AS HDAC INHIBITORS CRYSTAX PHARMACEUTICALS, S.L. (ES) 2010-06-24 WO disclosed