SCHEMBL3470387

SCHEMBL3470387

Cc1nn(C)c2nc(=O)n(-c3ccccc3)c(=O)c-2[n+]1[O-]

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 8/20 0.52
KDM4C Q9H3R0 4/20 0.41
RAF1 P04049 1/20 0.41
MAP2K1 Q02750 1/20 0.41
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
GSR P00390 1/20 0.40
CASP7 P55210 2/20 0.39
CASP6 P55212 2/20 0.39
NSD2 O96028 1/20 0.39
IDO1 P14902 1/20 0.39
CRHBP P24387 1/20 0.39
TDO2 P48775 1/20 0.39
CRHR2 Q13324 1/20 0.39
GAA P10253 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
APAF1 O14727 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3474651 0.77 TDP2 (0.47) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3471027 0.72 TDP2 (0.62) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3471238 0.72 TDP2 (0.80) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3476272 0.70 TDP2 (0.40) TDP2ALDH1A1KDM4EMAPTCRHBP
SCHEMBL3471243 0.69 HSF1 (0.42) TDP2ALDH1A1KDM4EMAPTCASP6
SCHEMBL3473639 0.68 TDP2 (0.58) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3475005 0.68 TDP2 (0.56) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3472489 0.68 TDP2 (0.57) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3471919 0.67 TDP2 (0.75) TDP2KDM4CRAF1MAP2K1ALDH1A1
SCHEMBL3472457 0.64 TDP2 (0.40) TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO claimed
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed