SCHEMBL3471919

SCHEMBL3471919

Cn1nc(Cc2ccccc2)nc2c(=O)n(-c3ccccc3)c(=O)nc1-2

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 11/20 0.75
KDM4C Q9H3R0 4/20 0.75
CASP6 P55212 3/20 0.47
CASP7 P55210 2/20 0.47
NSD2 O96028 1/20 0.47
IDO1 P14902 1/20 0.47
CRHBP P24387 1/20 0.47
TDO2 P48775 1/20 0.47
CRHR2 Q13324 1/20 0.47
KDM4E B2RXH2 3/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
RAF1 P04049 1/20 0.45
MAP2K1 Q02750 1/20 0.45
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
POLB P06746 2/20 0.44
THRB P10828 2/20 0.44
HTT P42858 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13272610 0.86 TDP2 (1.00) TDP2KDM4CCASP6CASP7KDM4E
SCHEMBL3471027 0.81 TDP2 (0.62) TDP2KDM4CCASP6CASP7NSD2
SCHEMBL3471912 0.79 TDP2 (0.66) TDP2KDM4CCASP6CRHBPCRHR2
SCHEMBL3471238 0.78 TDP2 (0.80) TDP2KDM4CCASP7KDM4EMAPT
SCHEMBL3473639 0.77 TDP2 (0.58) TDP2KDM4CCASP6CASP7NSD2
SCHEMBL3474479 0.74 TDP2 (1.00) TDP2KDM4CCASP6CASP7KDM4E
SCHEMBL3471911 0.73 TDP2 (0.77) TDP2KDM4CCASP6CASP7KDM4E
SCHEMBL3471993 0.72 TDP2 (0.73) TDP2KDM4CCASP6CASP7KDM4E
SCHEMBL3475916 0.68 TDP2 (0.67) TDP2KDM4CKDM4EMAPTLMNA
SCHEMBL14020030 0.67 TDP2 (0.73) TDP2KDM4CCASP6CASP7KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed