SCHEMBL3470514

SCHEMBL3470514

CC(C)(C)OC(=O)CN1C(=O)CCc2cc(-c3cccc(C(F)(F)F)c3)ccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.46
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
CYP1A2 P05177 1/20 0.45
PARP10 Q53GL7 1/20 0.40
PARP11 Q9NR21 1/20 0.40
GRIN1 Q05586 3/20 0.40
GRIN2B Q13224 3/20 0.40
RXRA P19793 2/20 0.40
NR1H2 P55055 2/20 0.40
NR1H3 Q13133 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
MAPT P10636 2/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
CCKBR P32239 1/20 0.39
NOTUM Q6P988 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314291 0.92 BRD4 (0.42) METCYP11B1CYP11B2PARP10PARP11
SCHEMBL3306832 0.92 MET (0.47) METCYP11B1CYP11B2CYP1A2MAPT
SCHEMBL3306622 0.85 CYP11B1 (0.46) METCYP11B1CYP11B2CYP1A2PARP10
SCHEMBL3308636 0.84 MET (0.45) METCYP11B1CYP11B2CYP1A2MAPT
SCHEMBL14866024 0.83 MET (0.48) METCYP11B1CYP11B2CYP1A2MAPT
SCHEMBL3301564 0.81 MET (0.47) METCYP11B1CYP11B2CYP1A2MAPT
SCHEMBL3473348 0.81 MET (0.47) METCYP11B1CYP11B2CYP1A2MEN1
SCHEMBL30393232 0.80 CYP11B1 (0.41) METCYP11B1CYP11B2CYP1A2HRH3
SCHEMBL3308428 0.78 CYP11B1 (0.42) METCYP11B1CYP11B2KMT2AHDAC6
SCHEMBL14866213 0.78 CCKBR (0.48) METMAPTCCKBRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010074807-A1 3, 4-DIHYDROQUINOLIN-2 ( 1H ) -ONE DERIVATIVES AS SODIUM CHANNEL MODULATORS GILEAD PALO ALTO, INC. (US) 2010-07-01 WO disclosed