SCHEMBL3471256

SCHEMBL3471256

Cn1nc(-c2cccs2)[n+]([O-])c2c(=O)n(C)c(=O)nc1-2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSF1 Q00613 7/20 0.54
NPC1 O15118 4/20 0.47
RAF1 P04049 3/20 0.47
MAP2K1 Q02750 3/20 0.47
KDM4E B2RXH2 3/20 0.47
ALDH1A1 P00352 3/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 2/20 0.47
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
GALK1 P51570 2/20 0.47
BLM P54132 2/20 0.47
NPSR1 Q6W5P4 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MEN1 O00255 1/20 0.47
HSP90AA1 P07900 1/20 0.47
HSP90AB1 P08238 1/20 0.47
THRB P10828 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13492890 0.76 TDP2 (0.55) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3472208 0.73 RAF1 (0.74) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3472489 0.69 TDP2 (0.57) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3472094 0.69 TDP2 (0.43) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3472830 0.69 TDP2 (0.43) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3292113 0.67 HSF1 (0.69) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL13273085 0.66 HSF1 (0.40) HSF1NPC1RAF1MAP2K1RAB9A
SCHEMBL10195758 0.64 HSF1 (1.00) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL3473513 0.64 TDP2 (0.54) HSF1NPC1RAF1MAP2K1KDM4E
SCHEMBL9118620 0.64 ALDH1A1 (0.49) HSF1NPC1RAF1MAP2K1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO claimed
WO-2010072807-A2 INHIBITORS OF CYSTATHIONINE BETA SYNTHASE TO REDUCE THE NEUROTOXIC OVERPRODUCTION OF ENDOGENOUS HYDROGEN SULFIDE FONDATION JEROME LEJEUNE (FR) 2010-07-01 WO disclosed