Erythromycin

Erythromycin

SCHEMBL3473986

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nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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The experimentally established mechanism targets of Erythromycin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 2/20 0.95
ABCC4 O15439 1/20 0.95
CYP3A4 P08684 9/20 0.85
SLCO1B3 Q9NPD5 3/20 0.85
SLCO1B1 Q9Y6L6 3/20 0.85
USP2 O75604 3/20 0.85
MAPK1 P28482 2/20 0.85
MEN1 O00255 1/20 0.85
TP53 P04637 1/20 0.85
MAPT P10636 1/20 0.85
HPGD P15428 1/20 0.85
ALOX12 P18054 1/20 0.85
RECQL P46063 1/20 0.85
BLM P54132 1/20 0.85
KMT2A Q03164 1/20 0.85
HSD17B10 Q99714 1/20 0.85
KCNH2 Q12809 5/20 0.79
ABCB1 P08183 2/20 0.79
MLNR O43193 2/20 0.79
TSHR P16473 2/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Erythromycin SCHEMBL7597008 0.97 ABCB11 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin SCHEMBL7597003 0.97 ABCB11 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin SCHEMBL11319270 0.97 ABCB11 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin SCHEMBL11319266 0.97 ABCB11 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Clarithromycin SCHEMBL7596572 0.94 ABCB11 (0.94) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Clarithromycin SCHEMBL7596567 0.94 ABCB11 (0.94) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin Propionate SCHEMBL25223334 0.92 CYP3A4 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin Propionate SCHEMBL29400629 0.92 CYP3A4 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin Propionate SCHEMBL3331 0.92 CYP3A4 (1.00) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1
Erythromycin SCHEMBL28256019 0.92 ABCB11 (0.86) ABCB11ABCC4CYP3A4SLCO1B3SLCO1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 264 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108379087-A Filling paste for dental pulp conservation treatment and preparation method thereof 徐崇明 2018-08-10 CN claimed
CN-107441501-A Drug-loaded liposome of antibacterial peptide modification and its production and use 四川大学 2017-12-08 CN claimed
CN-107446019-A Antibacterial peptide derivative and application thereof 四川大学 2017-12-08 CN claimed
CN-107320727-A Antibacterial peptide and antibiotic combinations antibacterials and its application method 四川大学 2017-11-07 CN claimed
CN-105492005-A Methods of treating microbial infections including mastitis LUODA PHARMA PTY LTD 2016-04-13 CN claimed
CN-105492004-A Method of treating topical microbial infections LUODA PHARMA PTY LTD 2016-04-13 CN claimed
CN-103705988-B A kind of intramedullary pin with multi-functional coatings and preparation method thereof SHANGHAI MICROPORT ORTHOPEDICS CO., LTD. (CN) 2016-02-17 CN claimed
CN-103705988-A Intramedullary nail having multifunctional coating and preparation method SHANGHAI MICROPORT ORTHOPEDICS 2014-04-09 CN claimed
US-20100221245-A1 TOPICAL SKIN CARE COMPOSITION DERMADOCTOR, LLC 2010-09-02 US claimed
CN-101039668-A Pharmaceutical formulations comprising an antibiotic, a triazole and a corticosteroid SCHERING PLOUGH LTD (CH) 2007-09-19 CN claimed
CN-1084631-C Powder medicine made of Chinese and Western medicines for treating toothache and preparation process thereof ZHANG CHANGLIANG (CN) 2002-05-15 CN claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
CN-1285220-A Powder medicine made of Chinese and Western medicines for treating toothache and preparation process thereof ZHANG CHANGLIANG (CN) 2001-02-28 CN claimed
CN-1031326-A Method with haloplankton as living drug carrier control fish and shrimp diseases QINGDAO OCEAN UNIVERSITY (CN) 1989-03-01 CN claimed
EP-3897452-B1 RESORBABLE NONWOVEN POUCHES FOR MEDICAL DEVICE IMPLANTS TEPHA INC (US) 2024-07-03 EP disclosed
US-20230201610-A1 RESORBABLE NONWOVEN POUCHES FOR MEDICAL DEVICE IMPLANTS TEPHA, INC. (US) 2023-06-29 US disclosed
US-11612754-B2 Resorbable nonwoven pouches for medical device implants TEPHA, INC. (US) 2023-03-28 US disclosed
US-4539234-A Urethral catheter capable of preventing urinary tract infection and process for producing the same UNITIKA LTD. (JP) 1985-09-03 US disclosed
US-4335115-A ERYTHROMYCIN, GLYCEROL MONOOLEATE, ETHANOL, AND ISOPROPYL MYRISTATE THE PROCTER & GAMBLE COMPANY (US) 1982-06-15 US disclosed
US-4102806-A DISPERSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1978-07-25 US disclosed