SCHEMBL3476295

SCHEMBL3476295

O=C(Nc1cc(C(F)(F)F)ccn1)c1cccnc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.67
MEN1 O00255 1/20 0.67
KMT2A Q03164 1/20 0.67
ALOX15 P16050 1/20 0.65
CASP1 P29466 1/20 0.65
NPSR1 Q6W5P4 1/20 0.65
HSD17B10 Q99714 1/20 0.65
MAPK8 P45983 1/20 0.58
MAPK10 P53779 1/20 0.58
DYRK1A Q13627 1/20 0.57
GRM5 P41594 1/20 0.56
RXFP1 Q9HBX9 1/20 0.56
TRPA1 O75762 1/20 0.55
CSF1R P07333 2/20 0.55
BRAF P15056 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.53
POLB P06746 1/20 0.53
TP53 P04637 2/20 0.52
NPC1 O15118 1/20 0.52
RAB9A P51151 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1968503 0.86 ALOX15 (0.60) TSHRALOX15CASP1NPSR1HSD17B10
Formic Acid SCHEMBL30595912 0.82 ALOX15 (0.55) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL15904287 0.82 TSHR (0.62) TSHRMEN1KMT2AALOX15CASP1
SCHEMBL30362452 0.82 TSHR (0.62) TSHRMEN1KMT2AALOX15CASP1
SCHEMBL15903185 0.81 ALOX15 (0.60) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL22243546 0.81 ALOX15 (0.60) TSHRALOX15CASP1NPSR1HSD17B10
SCHEMBL30643204 0.81 GRM5 (0.62) TSHRMEN1KMT2AALOX15CASP1
SCHEMBL5178391 0.80 MEN1 (1.00) TSHRMEN1KMT2ARXFP1TRPA1
SCHEMBL23015752 0.80 RAB9A (0.67) KMT2AHSD17B10MAPK8MAPK10SMN1; SMN2
SCHEMBL23410523 0.80 MAPK8 (0.62) HSD17B10MAPK8MAPK10GRM5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010034838-A2 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-04-01 WO claimed