SCHEMBL3477573

SCHEMBL3477573

CN(CCNc1cc(N2CCCC2)nc(N2CCCC2)n1)CCNc1ncnc2ncn(Cc3ccccc3)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 3/20 0.41
CASP5 P51878 3/20 0.41
SENP6 Q9GZR1 4/20 0.39
SENP7 Q9BQF6 3/20 0.39
APAF1 O14727 2/20 0.39
MAPT P10636 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ACHE P22303 2/20 0.38
HRH4 Q9H3N8 3/20 0.37
HRH1 P35367 1/20 0.36
CASP4 P49662 2/20 0.36
GBA1 P04062 1/20 0.36
CDK9 P50750 1/20 0.35
GALR2 O43603 1/20 0.35
GALR1 P47211 1/20 0.35
HTT P42858 2/20 0.35
POLB P06746 1/20 0.35
SENP8 Q96LD8 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NSD2 O96028 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3476226 0.87 HTT (0.51) CASP1CASP5MAPTHRH4HTT
SCHEMBL3475816 0.76 HRH4 (0.46) CASP1CASP5SENP6SENP7APAF1
SCHEMBL3476877 0.76 PIK3CD (0.45) MAPTSMN1; SMN2HTTLMNATDP1
SCHEMBL3474881 0.75 CYP2C19 (0.49) CASP1CASP5SENP6SENP7APAF1
SCHEMBL3477066 0.75 HRH4 (0.41) CASP1CASP5SENP6SENP7APAF1
SCHEMBL3477496 0.74 CDK1 (0.39) SENP6SENP7APAF1MAPTSMN1; SMN2
SCHEMBL2772821 0.73 SENP6 (0.48) CASP1CASP5SENP6SENP7APAF1
SCHEMBL3478373 0.73 HDAC1 (0.42) CASP1CASP5SENP6SENP7APAF1
SCHEMBL3476221 0.73 SENP6 (0.41) CASP1CASP5SENP6SENP7APAF1
SCHEMBL2773055 0.73 SENP6 (0.49) CASP1CASP5SENP6SENP7APAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010130900-A2 TRIAMINOPYRIMIDINE DERIVATIVES AS CDC25 PHOSPHATASE INHIBITORS IPSEN PHARMA S.A.S. (FR) 2010-11-18 WO claimed
WO-2010130900-A2 TRIAMINOPYRIMIDINE DERIVATIVES AS CDC25 PHOSPHATASE INHIBITORS IPSEN PHARMA S.A.S. (FR) 2010-11-18 WO disclosed