SCHEMBL3477845

SCHEMBL3477845

CC(C)(C)Cc1c[nH]c(-c2cccnc2F)c1F

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36
GPR84 Q9NQS5 1/20 0.33
TDO2 P48775 1/20 0.33
MAPT P10636 3/20 0.32
BRAF P15056 1/20 0.32
NPC1 O15118 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP3A4 P08684 1/20 0.30
CYP11B2 P19099 1/20 0.30
CASP6 P55212 1/20 0.30
MET P08581 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14899993 0.84 GPR84 (0.36) ALOX5APFEN1GPR84TDO2MAPT
SCHEMBL12417811 0.81 GPR84 (0.39) GPR84TDO2MAPTNPC1HTT
SCHEMBL12417843 0.80 GPR84 (0.40) GPR84TDO2MAPTCYP3A4CYP11B2
SCHEMBL1830980 0.78 NAPRT (0.33)
SCHEMBL2194154 0.76 NAPRT (0.38) MAPT
SCHEMBL1830977 0.76 SSTR4 (0.38)
SCHEMBL4566391 0.75 CHRM2 (0.32) NPC1HTT
SCHEMBL9969425 0.74 NPC1 (0.38) ALOX5APFEN1MAPTNPC1HTT
SCHEMBL3477844 0.74 TDO2 (0.33) TDO2MAPTCYP11B2
SCHEMBL1830978 0.74 DYRK1A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010024451-A1 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-03-04 WO disclosed