SCHEMBL34784

SCHEMBL34784

O=C(O)[C@@H](CS)C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.48
CPA3 P15088 1/20 0.48
CYP1A2 P05177 1/20 0.41
KIF11 P52732 3/20 0.41
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785507 1.00 FOLH1 (0.48) FOLH1CPA3CYP1A2KIF11CYP2C19
SCHEMBL11267940 0.88 CHRM2 (0.43) FOLH1CPA3CYP1A2CYP2C19TSHR
SCHEMBL11245351 0.85 FOLH1 (0.42) FOLH1CPA3CYP1A2KIF11CYP2C19
SCHEMBL1160457 0.80 FOLH1 (0.49) FOLH1CPA3KIF11
SCHEMBL17913818 0.80 FOLH1 (0.49) FOLH1CPA3KIF11
SCHEMBL7828921 0.79 ANPEP (0.52) FOLH1CPA3KIF11
SCHEMBL27346918 0.76 TSHR (0.47) CYP1A2KIF11CYP2C19TSHR
SCHEMBL4797477 0.76 KIF11 (0.53) KIF11
SCHEMBL27349964 0.76 TSHR (0.47) CYP1A2KIF11CYP2C19TSHR
SCHEMBL3185210 0.73 CYP2C19 (0.40) CYP1A2KIF11CYP2C19HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025027389-A1 BIOLOGICALLY ACTIVE COMPOUNDS COMPRISING A STAPLED OR STITCHED PEPTIDE SUTURA THERAPEUTICS LIMITED (GB) 2025-02-06 WO claimed
US-20250127797-A1 PRODRUG COMPRISING A DRUG-LINKER CONJUGATE ASCENDIS PHARMA A/S (DK) 2025-04-24 US disclosed
WO-2025027389-A1 BIOLOGICALLY ACTIVE COMPOUNDS COMPRISING A STAPLED OR STITCHED PEPTIDE SUTURA THERAPEUTICS LIMITED (GB) 2025-02-06 WO disclosed
US-11965851-B2 Grid coatings for capture of proteins and other compounds PURDUE RESEARCH FOUNDATION (US) 2024-04-23 US disclosed
WO-2024069229-A2 BIOLOGICALLY ACTIVE COMPOUNDS SUTURA THERAPEUTICS LTD (GB) 2024-04-04 WO disclosed
US-20240041897-A1 PRODRUG COMPRISING A DRUG LINKER CONJUGATE ASCENDIS PHARMA GMBH (DE) 2024-02-08 US disclosed
US-20220331334-A1 Prodrug Comprising a Drug-Linker Conjugate ASCENDIS PHARMA A/S (DK) 2022-10-20 US disclosed
US-11458212-B2 Molecular imaging of cancer cells in vivo H. LEE MOFFITT CANCER CENTER AND RESEARCH INSTITUTE, INC. (US) 2022-10-04 US disclosed
US-11458206-B2 Targeted conjugates and particles and formulations thereof TVA (ABC), LLC (US) 2022-10-04 US disclosed
US-20220288229-A1 TARGETED CONJUGATES ENCAPSULATED IN PARTICLES AND FORMULATIONS THEREOF TVA (ABC), LLC 2022-09-15 US disclosed
US-20050256301-A1 Cyclised conotoxin peptides THE UNIVERSITY OF QUEENSLAND (AU) 2005-11-17 US disclosed
EP-0618221-A2 Heterocyclic inhibitors of farnesyl protein transferase BRISTOL-MYERS SQUIBB COMPANY (US) 1994-10-05 EP disclosed
EP-0013261-B1 GUAIACOL ESTERS OF ALPHA- AND BETA-MERCAPTOPROPIONYLALANINE AND ALPHA- AND BETA-MERCAPTOPROPIONYLGLYCINE, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1982-12-01 EP disclosed
US-4350628-A OXIDATIVE DEHYDROGENATION WITH A BENZOQUINONE RESEARCH CORPORATION (US) 1982-09-21 US disclosed
US-4299842-A TREATMENT OF RESPIRATORY SYSTEM DISORDERS, NUCOLYTIC AGENTS CAVAZZA CLAUDIO 1981-11-10 US disclosed
US-4283328-A TREATING AN N-BLOCKED AMINO ACID RESIDUE WITH A TETRAMETHYL GUANIDINIUM SALT OF A PEPTIDE CHAIN RESEARCH CORPORATION (US) 1981-08-11 US disclosed
US-4261884-A DESIRABLE BIOLOGICAL PROPERTIES AND STABILITY TO ENZYME CLEAVAGE RESEARCH CORPORATION (US) 1981-04-14 US disclosed
EP-0013261-A1 Guaiacol esters of alpha- and beta-mercaptopropionylalanine and alpha- and beta-mercaptopropionylglycine, process for their preparation and pharmaceutical compositions containing same Sigma-Tau Industrie Farmaceutiche Riunite S.p.A. (IT) 1980-07-09 EP disclosed
EP-0010830-A2 Dehydropeptides Research Corporation (US) 1980-05-14 EP disclosed
US-4113714-A GROWTH HORMONE RELEASE INHIBITING UNDECAPEPTIDE AMERICAN HOME PRODUCTS CORPORATION (US) 1978-09-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220288229-A1 TARGETED CONJUGATES ENCAPSULATED IN PARTICLES AND FORMULATIONS THEREOF CD47, CD44, FURIN FOLH1 11/4885CPA3 100/4885CYP1A2 3115/4885
US-20050256301-A1 Cyclised conotoxin peptides VIP, CANX, IAPP FOLH1 1079/4885CPA3 29/4885CYP1A2 2114/4885
US-11458212-B2 Molecular imaging of cancer cells in vivo MKI67, ANXA4, ANXA3 FOLH1 17/4885CPA3 575/4885CYP1A2 4882/4885
US-11965851-B2 Grid coatings for capture of proteins and other compounds CD2BP2, CDC37, CD68 FOLH1 1417/4885CPA3 2650/4885CYP1A2 4501/4885
US-20240041897-A1 PRODRUG COMPRISING A DRUG LINKER CONJUGATE H1-0, H1-3, H1-2 FOLH1 651/4885CPA3 627/4885CYP1A2 262/4885
US-20220331334-A1 Prodrug Comprising a Drug-Linker Conjugate H1-0, H1-3, DLST FOLH1 620/4885CPA3 693/4885CYP1A2 263/4885
US-20250127797-A1 PRODRUG COMPRISING A DRUG-LINKER CONJUGATE H1-0, H1-3, DLST FOLH1 620/4885CPA3 693/4885CYP1A2 263/4885
US-11458206-B2 Targeted conjugates and particles and formulations thereof SSTR5, SSTR1, SSTR4 FOLH1 54/4885CPA3 48/4885CYP1A2 4323/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.