SCHEMBL3485840

SCHEMBL3485840

COC(=O)C(NC=O)C(C)O

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 3/20 0.41
CA12 O43570 2/20 0.41
ADH1B P00325 1/20 0.39
ADH1C P00326 1/20 0.39
ADH1A P07327 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.37
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
KMT2A Q03164 2/20 0.32
TSHR P16473 3/20 0.32
MEN1 O00255 1/20 0.32
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693398 1.00 CA14 (0.41) CA14CA12ADH1BADH1CADH1A
SCHEMBL3201079 0.84 CA14 (0.52) CA14CA12ADH1BADH1CADH1A
SCHEMBL8610890 0.84 CA14 (0.52) CA14CA12ADH1BADH1CADH1A
SCHEMBL27600917 0.80 ADH1B (0.33) CA14CA12ADH1BADH1CADH1A
SCHEMBL8017539 0.78 NOS3 (0.43) TAS1R3TAS1R1
SCHEMBL31509428 0.78 NOS3 (0.43) TAS1R3TAS1R1
SCHEMBL18823490 0.77 ADH1B (0.42) ADH1BADH1CADH1AKMT2AMEN1
SCHEMBL18712598 0.77 ADH1B (0.42) ADH1BADH1CADH1AKMT2AMEN1
SCHEMBL22166168 0.77 ADH1B (0.42) ADH1BADH1CADH1AKMT2AMEN1
SCHEMBL17313812 0.77 ADH1B (0.42) ADH1BADH1CADH1AKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130184462-A1 METHOD FOR PREDICTING AND MODELING ANTI-PSYCHOTIC ACTIVITY USING VIRTUAL SCREENING MODEL COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2013-07-18 US disclosed
US-20100029724-A1 SCREENING METHOD TAKEDA PHARMACEUTICAL COMPANY LIMITED 2010-02-04 US disclosed
EP-2039779-A1 SCREENING METHOD Takeda Pharmaceutical Company Limited (JP) 2009-03-25 EP disclosed
US-20080287438-A1 Agent for preventing or treating neuropathy MOMOSE YU 2008-11-20 US disclosed
US-7423159-B2 Agent for preventing or treating neuropathy TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-09 US disclosed
US-7183276-B2 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-02-27 US disclosed
US-20060004069-A1 Agent for preventing or treating neuropathy TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-05 US disclosed
US-20050090534-A1 Azole compounds TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-04-28 US disclosed
EP-1486490-A1 AZOLE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2004-12-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050090534-A1 Azole compounds AHR, NR0B2, NR2C2 CA14 2335/4885CA12 2146/4885ADH1B 252/4885
US-20100029724-A1 SCREENING METHOD NR2C2, NCOR2, NCOA2 CA14 1529/4885CA12 723/4885ADH1B 497/4885
US-20060004069-A1 Agent for preventing or treating neuropathy NR2C2, NR0B2, NR2E1 CA14 4354/4885CA12 3141/4885ADH1B 699/4885
US-20080287438-A1 Agent for preventing or treating neuropathy NR2C2, NR0B2, NR2E1 CA14 4354/4885CA12 3141/4885ADH1B 699/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.