SCHEMBL3492877

SCHEMBL3492877

Cc1ccc2c(c1)C(=O)CC1(CCN(C(=O)c3c(N)sc4ncccc34)CC1)S2

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.33
ACACB O00763 6/20 0.33
ACACA Q13085 3/20 0.33
CYP46A1 Q9Y6A2 3/20 0.33
KMT2A Q03164 3/20 0.32
MEN1 O00255 2/20 0.32
IKBKB O14920 1/20 0.32
CHUK O15111 1/20 0.32
LIMK1 P53667 1/20 0.32
NPC1 O15118 3/20 0.32
USP2 O75604 2/20 0.32
TP53 P04637 2/20 0.32
RAB9A P51151 2/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
OPRD1 P41143 1/20 0.31
CES2 O00748 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3490756 0.88 NPC1 (0.35) ACACBACACAKMT2AMEN1IKBKB
SCHEMBL3490730 0.88 ACACB (0.40) ATMACACBACACACYP46A1KMT2A
SCHEMBL3490732 0.88 ACACB (0.40) ATMACACBACACACYP46A1KMT2A
SCHEMBL3493749 0.87 SLC6A7 (0.32) ACACBACACAIKBKBCHUKLIMK1
SCHEMBL3494669 0.87 ACACB (0.40) ATMACACBACACACYP46A1KMT2A
SCHEMBL3494665 0.87 ACACB (0.40) ATMACACBACACACYP46A1KMT2A
SCHEMBL3493125 0.84 PDE4B (0.33) ACACBACACAKMT2AMEN1NPC1
SCHEMBL3492830 0.83 ACACB (0.52) ACACBACACA
SCHEMBL3492828 0.83 ACACB (0.52) ACACBACACA
SCHEMBL13340541 0.82 ACACB (0.39) ATMACACBACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100113418-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-06 US disclosed
US-20100113418-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-06 US disclosed
US-20100113418-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-06 US disclosed
EP-2123652-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-11-25 EP disclosed
EP-2123652-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2009-11-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113418-A1 HETEROCYCLIC COMPOUND ACACA, ACAT1, CPT1B ATM 622/4885ACACB 5/4885ACACA 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.