SCHEMBL3499819

SCHEMBL3499819

CCOC(=O)C1(N)Cc2ccc(-c3ccc(F)c(Cl)c3)cc2C1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.44
ICMT O60725 5/20 0.38
PGR P06401 3/20 0.38
SLC1A3 P43003 1/20 0.38
SLC1A2 P43004 1/20 0.38
SLC1A1 P43005 1/20 0.38
APP P05067 1/20 0.37
BACE1 P56817 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
PTPRC P08575 1/20 0.37
PTPN2 P17706 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPA Q15257 1/20 0.37
KMT2A Q03164 2/20 0.37
MEN1 O00255 1/20 0.37
ERCC1 P07992 1/20 0.36
ERCC4 Q92889 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3498220 0.88 MEN1 (0.45) TDP2KMT2AMEN1OPRM1
Hydrochloric Acid SCHEMBL3498072 0.87 OPRM1 (0.45) TDP2KMT2AMEN1OPRM1
SCHEMBL3499676 0.85 OPRM1 (0.43) PTGS2KMT2AMEN1OPRM1
SCHEMBL3498275 0.83 OPRM1 (0.41) ICMTOPRM1
SCHEMBL13328485 0.82 MEN1 (0.46) KMT2AMEN1OPRM1
SCHEMBL3305558 0.80 OPRM1 (0.44) KMT2AMEN1OPRM1
Hydrochloric Acid SCHEMBL3498150 0.80 GRIA1 (0.41) KMT2AMEN1OPRM1
SCHEMBL13328476 0.79 OPRM1 (0.45) KMT2AMEN1OPRM1
SCHEMBL3311022 0.79 OPRM1 (0.39) KMT2AMEN1OPRM1
SCHEMBL3499699 0.79 AOC3 (0.42) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100130737-A1 Regulating Agent of GPR34 Receptor Function TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-27 US disclosed
US-20100130737-A1 Regulating Agent of GPR34 Receptor Function TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-27 US disclosed
US-20100130737-A1 Regulating Agent of GPR34 Receptor Function TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-05-27 US disclosed
EP-1849465-A1 AGENT FOR CONTROLLING FUNCTION OF GPR34 RECEPTOR Takeda Pharmaceutical Company Limited (JP) 2007-10-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100130737-A1 Regulating Agent of GPR34 Receptor Function GPR34, GPR4, GPR6 TDP2 4872/4885ICMT 4502/4885PGR 233/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.