Fludarabine

Fludarabine

SCHEMBL3510

Nc1nc(F)nc2c1ncn2[C@@H]1O[C@H](CO)[C@@H](O)[C@@H]1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 1.00
NT5E P21589 1/20 1.00
HIF1A Q16665 1/20 1.00
ADORA2A P29274 7/20 0.73
ADORA2B P29275 5/20 0.73
ADORA3 P0DMS8 3/20 0.71
CA5A P35218 1/20 0.70
ADORA1 P30542 2/20 0.69
DPP4 P27487 1/20 0.69
MEN1 O00255 1/20 0.69
SLC28A1 O00337 1/20 0.69
MAP3K7 O43318 1/20 0.69
SLC28A2 O43868 1/20 0.69
GAPDH P04406 1/20 0.69
MAPK1 P28482 1/20 0.69
STAT6 P42226 1/20 0.69
PI4KA P42356 1/20 0.69
KMT2A Q03164 1/20 0.69
SMN1; SMN2 Q16637 1/20 0.69
PI4K2B Q8TCG2 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fludarabine SCHEMBL3047091 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL12018219 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL12018226 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL3655059 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL13046076 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL977919 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL12232219 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL13046078 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL14031844 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B
Fludarabine SCHEMBL12019517 1.00 LMNA (1.00) LMNANT5EHIF1AADORA2AADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 110634 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12584903-B2 Cellular-based method for determining the potency of defibrotide GENTIUM S.R.L. (IT) 2026-03-24 US claimed
WO-2025111589-A1 COMPOSITIONS AND METHODS FOR ENHANCING DRUG RESISTANCE IN CELLS MEDICI THERAPEUTICS, INC. (US) 2025-05-30 WO claimed
US-12042480-B2 Methods, agents, and compositions for the treatment of acute myeloid leukemia UNIVERSITY OF CINCINNATI (US) 2024-07-23 US claimed
US-12042542-B2 Synthetic antibody mimetic compounds (SYAMS) targeting cancer, especially prostate cancer YALE UNIVERSITY (US) 2024-07-23 US claimed
US-20240238291-A1 COMBINATIONS FOR TREATMENT OF CANCER SYNDAX PHARMACEUTICALS INC (US) 2024-07-18 US claimed
WO-2024002154-A9 ANTI-FGFR3 ANTIBODY CONJUGATE AND MEDICAL USE THEREOF GENEQUANTUM HEALTHCARE (SUZHOU) CO., LTD. (CN) 2024-07-18 WO claimed
US-20240238282-A1 METHODS OF TREATING CANCER AND ISCHEMIA DISEASES BY INHIBITION AND INTERVENTION OF ATR PROLYL ISOMERIZATION THE UNIVERSITY OF TOLEDO (US) 2024-07-18 US claimed
US-20240239799-A1 (S)-1-(5-((PYRIDIN-3-YL)THIO)PYRAZIN-2-YL)-4'H,6'H-SPIRO[PIPERIDINE-4,5'-PYRROLO [1,2-B]PYRAZOL]-4'-AMINE DERIVATIVES AND SIMILAR COMPOUNDS AS SHP2 INHIBITORS FOR THE TREATMENT OF E.G. CANCER C.N.C.C.S. S.C.A.R.L. COLLEZIONE NAZIONALE DEI COMPOSTI CHIMICI E CENTRO SCREENING (IT) 2024-07-18 US claimed
WO-2024152052-A1 COMPOSITIONS COMPRISING FLUDARABINE PHOSPHATE AND METHODS OF MAKING AND USING SAME TO TREAT CANCER AREVA PHARMACEUTICALS INC. (US) 2024-07-18 WO claimed
US-20240240146-A1 PROCESSES FOR PRODUCTION OF TUMOR INFILTRATING LYMPHOCYTES AND USES OF THE SAME IN IMMUNOTHERAPY IOVANCE BIOTHERAPEUTICS, INC. 2024-07-18 US claimed
WO-1996032115-A1 A PHARMACEUTICAL COMPOSITION CONTAINING N-PHOSPHONOGLYCINE DERIVATIVES FOR INHIBITING THE GROWTH OF VIRUSES AND CANCERS THE PROCTER & GAMBLE COMPANY (US) 1996-10-17 WO claimed
EP-0670845-A1 PROCESS FOR THE PREPARATION OF FLUDARABINE PHOSPHATE FROM GUANOSINE SCHERING AKTIENGESELLSCHAFT (DE) 1995-09-13 EP claimed
WO-1994012514-A1 PROCESS FOR THE PREPARATION OF FLUDARABINE PHOSPHATE FROM GUANOSINE SCHERING AKTIENGESELLSCHAFT (DE) 1994-06-09 WO claimed
US-5296589-A Dissolving in nonreactive solvent, reacting with hydrogen, palladium chloride, hydrochloric acid in sealed vessel at elevated pressure, removing palladium chloride, neutralizing, separating product ASH STEVENS, INC. (US) 1994-03-22 US claimed
EP-0359347-B1 COVALENTLY-LINKED COMPLEXES AND METHODS FOR ENHANCED CYTOTOXICITY AND IMAGING NEORX CORPORATION (US) 1992-12-23 EP claimed
US-5159067-A 5'-Diphosphohexose nucleoside pharmaceutical compositions UNIVERSITY OF GEORGIA RESEARCH FOUNDATION INC. (US) 1992-10-27 US claimed
WO-1991000867-A1 5'-DIPHOSPHOHEXOSE NUCLEOSIDE PHARMACEUTICAL COMPOSITIONS UNIVERSITY OF GEORGIA RESEARCH FOUNDATION, INC. (US) 1991-01-24 WO claimed
US-4357324-A Prodrug derivatives of 9β-D-arabinofuranosyl-2-fluoroadenine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1982-11-02 US claimed
US-4210745-A Procedure for the preparation of 9-β-D-arabinofuranosyl-2-fluoroadenine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1980-07-01 US claimed
US-4188378-A Anticancer and antiviral activity of 9-β-D-arabinofuranosyl-2-fluoroadenine THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH, EDUCATION AND WELFARE (US) 1980-02-12 US claimed