SCHEMBL3525528

SCHEMBL3525528

COCCN1C(=O)c2c(O)c(=O)c(C(=O)NCc3ccccc3OC)cn2CC1O

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.50
HPGD P15428 1/20 0.46
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
F2 P00734 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
POLB P06746 1/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2186099 0.93 TP53 (0.43) MEN1KMT2ASMN1; SMN2POLBTP53
SCHEMBL2187373 0.91 SLC22A2 (0.43) MAPK1
SCHEMBL3529763 0.91 SLC22A2 (0.43)
SCHEMBL2186319 0.90 SLC22A2 (0.53)
SCHEMBL2185991 0.89 SLC22A2 (0.44)
SCHEMBL3528388 0.87 P2RX7 (0.50)
SCHEMBL2185556 0.86
SCHEMBL2187402 0.85 SLC22A2 (0.54)
SCHEMBL2186875 0.85 SLC22A2 (0.62)
SCHEMBL3528016 0.84 ALDH1A1 (0.43) MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7858788-B2 Bicyclic carbamoylpyridone derivative having HIV integrase inhibitory activity SHIONOGI & CO., LTD. (JP) 2010-12-28 US disclosed
EP-1852434-A1 BICYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITING ACTIVITY Shionogi Co., Ltd. (JP) 2007-11-07 EP disclosed