Ilomastat

Ilomastat

SCHEMBL35303

CNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](CC(=O)NO)CC(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 16/20 1.00
MMP9 P14780 16/20 1.00
MMP8 P22894 14/20 1.00
MMP1 P03956 7/20 1.00
MMP3 P08254 3/20 1.00
MMP14 P50281 2/20 1.00
ADAM10 O14672 1/20 1.00
ADAM12 O43184 1/20 1.00
ADAMTS4 O75173 1/20 1.00
MMP7 P09237 1/20 1.00
MMP12 P39900 1/20 1.00
MMP13 P45452 1/20 1.00
MMP15 P51511 1/20 1.00
MMP16 P51512 1/20 1.00
ADAM17 P78536 1/20 1.00
ADAM9 Q13443 1/20 1.00
MMP26 Q9NRE1 1/20 1.00
MMP17 Q9ULZ9 1/20 1.00
ADAMTS5 Q9UNA0 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ilomastat SCHEMBL29412562 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL7870487 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL4394885 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL6691646 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL8190117 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL13575799 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
Ilomastat SCHEMBL4293696 1.00 MMP2 (1.00) MMP2MMP9MMP8MMP1MMP3
SCHEMBL8394283 0.92 MMP2 (0.85) MMP2MMP9MMP8MMP1MMP3
SCHEMBL4845965 0.91 MMP2 (0.84) MMP2MMP9MMP8MMP1MMP3
SCHEMBL5558468 0.90 MMP2 (0.82) MMP2MMP9MMP8MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12338 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20250360106-A1 PREVENTING IMMUNOTHERAPY-INDUCED EDEMA USING ANGIOTENSIN RECEPTOR BLOCKERS MASSACHUSETTS GEN HOSPITAL (US) 2025-11-27 US claimed
EP-4644418-A1 NANOBODY TARGETING BCMA, CHIMERIC ANTIGEN RECEPTOR AND USE THEREOF Hebei Senlang Biotechnology Co. Ltd. (CN) 2025-11-05 EP claimed
US-20250332225-A1 Injectable Neutral pH Collagen-Based Composition For Mesotherapy SHANGHAI QISHENG BIOLOGICAL PREPARATION CO LTD (CN) 2025-10-30 US claimed
US-20250262268-A1 Methods and Compositions for Inhibiting Viral Infection NEW YORK UNIVERSITY 2025-08-21 US claimed
US-20250221991-A1 COMBINATION THERAPY FOR THE TREATMENT OF CANCER METASTASES UNIVERSITY OF CINCINNATI (US) 2025-07-10 US claimed
CN-119955884-A Oat polypeptide extracted by directional enzyme digestion and method and application thereof 杭州恩和生物科技有限公司 2025-05-09 CN claimed
CN-119639852-A Preparation process and application of small fruit coffee grounds derived polypeptides 杭州恩和生物科技有限公司 2025-03-18 CN claimed
CN-117777290-B Monoclonal antibody specifically recognizing CLDN18.2 and related products, methods and uses thereof 深圳豪石生物科技有限公司 2025-01-24 CN claimed
JP-2000503660-A 2000-03-28 JP claimed
EP-0942746-A1 INHIBITION OF INVASIVE REMODELLING FONDEN TIL FREMME AF EKSPERIMENTEL CANCERFORSKNING (DK) 1999-09-22 EP claimed
US-5948780-A ADMINISTERING A METALLOPROTEINASE INHIBITOR WARNER-LAMBERT COMPANY (US) 1999-09-07 US claimed
EP-0883398-A4 METHOD OF INHIBITING PHOTOAGING OF SKIN UNIV MICHIGAN (US) 1999-05-12 EP claimed
CN-1211178-A Method for inhibiting skin photoaging UNIV MICHIGAN (US) 1999-03-17 CN claimed
EP-0883398-A1 METHOD OF INHIBITING PHOTOAGING OF SKIN THE UNIVERSITY OF MICHIGAN (US) 1998-12-16 EP claimed
US-5837224-A Method of inhibiting photoaging of skin THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 1998-11-17 US claimed
WO-1998025597-A2 METHOD FOR TREATING AND PREVENTING HEART FAILURE AND VENTRICULAR DILATATION WARNER-LAMBERT COMPANY (US) 1998-06-18 WO claimed
WO-1998024474-A1 INHIBITION OF INVASIVE REMODELLING FONDEN TIL FREMME AF EKSPERIMENTEL CANCERFORSKNING (DK) 1998-06-11 WO claimed
WO-1997025969-A1 METHOD OF INHIBITING PHOTOAGING OF SKIN THE UNIVERSITY OF MICHIGAN (US) 1997-07-24 WO claimed