SCHEMBL3534952

SCHEMBL3534952

CCOC(=O)CN(CCCCC(=O)O)Cc1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.54
ACHE P22303 1/20 0.54
HDAC3 O15379 2/20 0.50
HDAC1 Q13547 2/20 0.50
HDAC2 Q92769 2/20 0.50
HDAC8 Q9BY41 2/20 0.50
NCOR2 Q9Y618 2/20 0.50
LTA4H P09960 3/20 0.48
ALDH1A1 P00352 2/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
KDM4A O75164 2/20 0.47
KDM4C Q9H3R0 2/20 0.47
ALOX5 P09917 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.44
APP P05067 2/20 0.44
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27526991 0.99 BCHE (0.56) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL10848318 0.96 ALOX5 (0.51) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL5407867 0.93 BCHE (0.55) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL19533628 0.91 BCHE (0.53) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL29151455 0.91 ALOX5 (0.47) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL6659347 0.89 ALOX5 (0.59) BCHEACHEHDAC3HDAC1HDAC2
SCHEMBL4321470 0.86 SMN1; SMN2 (0.51) BCHEACHELTA4HALDH1A1MAPK1
SCHEMBL20506778 0.86 ALDH1A1 (0.49) BCHEACHELTA4HALDH1A1ALOX5
SCHEMBL3184733 0.86 ALDH1A1 (0.54) LTA4HALDH1A1ALOX5SMN1; SMN2LMNA
SCHEMBL31301745 0.86 ALOX5 (0.52) BCHEACHEHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112538084-B Novel KRAS G12C protein inhibitor and preparation method and application thereof 信达生物制药(苏州)有限公司 2023-06-20 CN disclosed
EP-3246317-B1 BTK INHIBITOR HUBEI BIO PHARMACEUTICAL INDUSTRIAL TECH INSTITUTE INC (CN) 2023-02-22 EP disclosed
CN-112538084-A Novel KRAS G12C protein inhibitor and preparation method and application thereof 信达生物制药(苏州)有限公司 2021-03-23 CN disclosed
US-7727979-B2 Guanidine derivatives and their use as neuropeptide FF receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2010-06-01 US disclosed
CN-100355758-C Guanidine derivatives and use thereof as neuropeptide FF receptor antagonists ACTELION PHARMACEUTICALS LTD (CH) 2007-12-19 CN disclosed
US-20060194788-A1 Guanidine derivatives and their use as neuropeptide ff receptor antagonists ACTELION PHARMACEUTICALS LTD. (CH) 2006-08-31 US disclosed
CN-1761673-A guanidine derivatives and their use as neuropeptide FF receptor antagonists ACTELION PHARMACEUTICALS LTD (CH) 2006-04-19 CN disclosed
EP-1608662-A1 GUANIDINE DERIVATIVES AND USE THEREOF AS NEUROPEPTIDE FF RECEPTOR ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2005-12-28 EP disclosed
WO-2004083218-A1 GUANIDINE DERIVATIVES AND USE THEREOF AS NEUROPEPTIDE FF RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2004-09-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060194788-A1 Guanidine derivatives and their use as neuropeptide ff receptor antagonists NPFFR1, OGFR, NPFFR2 BCHE 1147/4885ACHE 516/4885HDAC3 953/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.