SCHEMBL3535903

SCHEMBL3535903

CCN1CCN(c2ccc3nc(-c4n[nH]c5c(Cl)cccc45)n(C)c3c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 2/20 0.47
FGFR1 P11362 3/20 0.41
FGFR2 P21802 1/20 0.41
KHK P50053 2/20 0.41
HTR6 P50406 2/20 0.41
OPRM1 P35372 2/20 0.39
KDM4E B2RXH2 1/20 0.39
OPRD1 P41143 1/20 0.39
FLT1 P17948 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
WEE1 P30291 1/20 0.38
ADRA2A P08913 2/20 0.37
KDM1A O60341 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
GAA P10253 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
DRD4 P21917 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3542577 0.89 KHK (0.41) LCKFGFR1FGFR2KHKHTR6
SCHEMBL3539745 0.87 PRKDC (0.41) LCKFGFR1FGFR2KHKKDM4E
SCHEMBL3540020 0.85 LMNA (0.44) LCKFGFR1FGFR2KHKOPRM1
SCHEMBL3538529 0.84 FGFR1 (0.51) LCKFGFR1FGFR2KHKHTR6
SCHEMBL3537155 0.83 KHK (0.42) FGFR1FGFR2KHKHTR6FLT1
SCHEMBL3538866 0.80 FGFR1 (0.51) FGFR1FGFR2KHKHTR6KDM4E
SCHEMBL3537657 0.79 PRKDC (0.46) FGFR1FGFR2KHKKDM4EFLT1
SCHEMBL3534853 0.78 FGFR1 (0.48) FGFR1FGFR2KHKFLT1DRD4
SCHEMBL3536833 0.78 FGFR1 (0.48) FGFR1FGFR2KHKFLT1DRD4
SCHEMBL3534930 0.77 SMN1; SMN2 (0.45) FGFR1KDM4EMEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7642278-B2 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2010-01-05 US disclosed
US-7642278-B2 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2010-01-05 US disclosed
US-7642278-B2 Nitrogen compounds such as 3-(5-morpholin-4-yl-1H-benz-imidazol-2-yl)-1H-indazole and/or isomers, used as immunology modulators, antidiabetic agents, antiogenesis inhibitors or for prophylaxis of Alzheimer's disease NOVARTIS VACCINES AND DIAGNOSTICS, INC. (US) 2010-01-05 US disclosed
US-20060079564-A1 Indazole benzimidazole compounds CHIRON CORPORATION 2006-04-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079564-A1 Indazole benzimidazole compounds ABL1, ABL2, ALK LCK 51/4885FGFR1 886/4885FGFR2 1236/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.