SCHEMBL3537469

SCHEMBL3537469

COc1cc(Cl)ccc1OBOc1ccc(Cl)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.47
SLC6A4 P31645 5/20 0.44
SLC6A2 P23975 4/20 0.44
SLC6A3 Q01959 3/20 0.44
KCNH2 Q12809 1/20 0.44
TTR P02766 2/20 0.44
LMNA P02545 1/20 0.44
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TP53 P04637 1/20 0.41
HTR3E A5X5Y0 2/20 0.41
HTR3B O95264 2/20 0.41
HTR3A P46098 2/20 0.41
HTR3D Q70Z44 2/20 0.41
HTR3C Q8WXA8 2/20 0.41
ACHE P22303 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL519223 0.92 TRPV4 (0.47) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL29636402 0.84 TRPV4 (0.55) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL2127233 0.84 TRPV4 (0.55) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL15031545 0.84 TTR (0.46) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL28298273 0.82 TRPV4 (0.53) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL3411402 0.79 TSHR (0.49) SLC6A4SLC6A2ALDH1A1MEN1KMT2A
SCHEMBL19697763 0.77 TRPV4 (0.48) TRPV4SLC6A4SLC6A2SLC6A3KCNH2
SCHEMBL624403 0.77 TSHR (0.47) SLC6A4SLC6A2SLC6A3LMNAALDH1A1
SCHEMBL4289243 0.77 CYP3A4 (0.45) TRPV4SLC6A4KCNH2LMNAALDH1A1
SCHEMBL29273440 0.77 TRPV4 (0.48) TRPV4SLC6A4SLC6A2SLC6A3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645773-B2 Thiazoles as inhibitors of 11β-hydroxysteroid dehydrogenase HOFFMANN-LA ROCHE INC. (US) 2010-01-12 US disclosed