SCHEMBL519223

SCHEMBL519223

COc1ccc(Cl)cc1OBOc1cc(Cl)ccc1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.47
HTR3E A5X5Y0 2/20 0.44
HTR3B O95264 2/20 0.44
HTR3A P46098 2/20 0.44
HTR3D Q70Z44 2/20 0.44
HTR3C Q8WXA8 2/20 0.44
LMNA P02545 2/20 0.44
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TP53 P04637 1/20 0.41
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 2/20 0.41
KCNH2 Q12809 1/20 0.41
ACHE P22303 1/20 0.40
TTR P02766 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3537469 0.92 TRPV4 (0.47) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL29636402 0.84 TRPV4 (0.55) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL2127233 0.84 TRPV4 (0.55) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL15031950 0.84 HTR3E (0.45) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL28298273 0.82 TRPV4 (0.53) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL2477899 0.79 TSHR (0.49) ALDH1A1KDM4EMEN1KMT2ASLC6A2
SCHEMBL624403 0.77 TSHR (0.47) LMNAALDH1A1KDM4EMEN1KMT2A
SCHEMBL4289243 0.77 CYP3A4 (0.45) TRPV4LMNAALDH1A1SLC6A4KCNH2
SCHEMBL4350642 0.77 TRPV4 (0.48) TRPV4HTR3EHTR3BHTR3AHTR3D
SCHEMBL188251 0.77 ACHE (0.71) LMNAALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON INC (US) 2026-03-12 US disclosed
US-12509474-B2 Inhibitors of complement factors and uses thereof ANNEXON, INC. (US) 2025-12-30 US disclosed
US-12291502-B2 Topoisomerase II-alpha inhibitors and methods of treating cancer using the same THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2025-05-06 US disclosed
US-20240109920-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON, INC. 2024-04-04 US disclosed
US-11814404-B2 Inhibitors of complement factors and uses thereof ANNEXON, INC. (US) 2023-11-14 US disclosed
EP-4185592-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF Annexon, Inc. (US) 2023-05-31 EP disclosed
US-20230105776-A1 Topoisomerase II-alpha Inhibitors and Methods of Treating Cancer Using the Same UNITED STATES GOVERNMENT 2023-04-06 US disclosed
US-20220048930-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON, INC. 2022-02-17 US disclosed
WO-2020205991-A1 TOPOISOMERASE II-alpha INHIBITORS AND METHODS OF TREATING CANCER USING THE SAME THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE (US) 2020-10-08 WO disclosed
US-10246422-B2 Heterocyclic compounds and use thereof in medicine and in cosmetics GALDERMA RESEARCH & DEVELOPMENT (FR) 2019-04-02 US disclosed
US-20040204386-A1 Pyrimidines and uses thereof CELL THERAPEUTICS, INC. 2004-10-14 US disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2004016615-A1 PYRAZOLO (4,3c) CINNOLINE COMPOUNDS AS INHIBITORS OF ITK KINASE ACTIVITY ASTRAZENECA AB (SE) 2004-02-26 WO disclosed
US-20030225110-A1 Tetrahydroquinoline derivatives as antithrombotic agents BRISTOL-MYERS SQUIBB PHARMA COMPANY 2003-12-04 US disclosed
US-20030225042-A1 Antipicornaviral compounds and compositions, their uses, and materials for their synthesis JOHNSON THEODORE O (US) 2003-12-04 US disclosed
US-6610730-B2 Viricides; protease inbhibitor AGOURON PHARMACEUTICALS, INC. 2003-08-26 US disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed
EP-1274682-A2 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2003-01-15 EP disclosed
US-20020006943-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis AGOURON PHARMACEUTICALS, INC. 2002-01-17 US disclosed
WO-2001079167-A2 ANTIPICORNAVIRAL COMPOUNDS AND COMPOSITIONS, THEIR PHARMACEUTICAL USES, AND MATERIALS FOR THEIR SYNTHESIS AGOURON PHARMACEUTICALS, INC. (US) 2001-10-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (12 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030225110-A1 Tetrahydroquinoline derivatives as antithrombotic agents TFPI, TFPI2, SERPINC1 TRPV4 2159/4885HTR3E 1207/4885HTR3B 306/4885
US-20240109920-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFB, CFH, C9 TRPV4 4621/4885HTR3E 2568/4885HTR3B 1598/4885
US-20230105776-A1 Topoisomerase II-alpha Inhibitors and Methods of Treating Cancer Using the Same TOP2A, TOP1, TOP2B TRPV4 4557/4885HTR3E 4220/4885HTR3B 3890/4885
US-20040204386-A1 Pyrimidines and uses thereof LPCAT3, LPCAT1, APRT TRPV4 4456/4885HTR3E 3581/4885HTR3B 3310/4885
US-20220048930-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFB, CFH, C9 TRPV4 4621/4885HTR3E 2568/4885HTR3B 1598/4885
US-12291502-B2 Topoisomerase II-alpha inhibitors and methods of treating cancer using the same TOP2A, TOP1, TOP2B TRPV4 4557/4885HTR3E 4220/4885HTR3B 3890/4885
US-11814404-B2 Inhibitors of complement factors and uses thereof CFB, CFH, C9 TRPV4 4621/4885HTR3E 2568/4885HTR3B 1598/4885
US-12509474-B2 Inhibitors of complement factors and uses thereof SSB, UACA, CFH TRPV4 4840/4885HTR3E 2961/4885HTR3B 2988/4885
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFH, CFB, C5 TRPV4 4864/4885HTR3E 926/4885HTR3B 888/4885
US-10246422-B2 Heterocyclic compounds and use thereof in medicine and in cosmetics MC1R, BDKRB2, CCKBR TRPV4 159/4885HTR3E 188/4885HTR3B 144/4885
US-20030225042-A1 Antipicornaviral compounds and compositions, their uses, and materials for their synthesis RNASEL, SARNP, RNASEH1 TRPV4 4095/4885HTR3E 3632/4885HTR3B 4057/4885
US-20020006943-A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis PRCP, RNPEP, SERPINB1 TRPV4 3769/4885HTR3E 3310/4885HTR3B 3917/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.