SCHEMBL3540409

SCHEMBL3540409

Nc1cc(OBOc2ccc(Cl)c(N)c2)ccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.48
TP53 P04637 1/20 0.48
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
DRD4 P21917 1/20 0.41
GAA P10253 2/20 0.40
NR4A1 P22736 1/20 0.38
CYP3A4 P08684 3/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
TUBB2A Q13885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL177501 0.79 HSP90AA1 (0.47) TSHRTP53CYP3A4MEN1KMT2A
SCHEMBL110854 0.76 ALDH1A1 (0.57) TSHRTP53CA12CA1CA2
Hydrochloric Acid SCHEMBL414955 0.74 ALDH1A1 (0.61) TSHRTP53CA12CA1CA2
SCHEMBL1124557 0.74 ALDH1A1 (0.48) TSHRGAANR4A1CYP3A4TUBB4A
SCHEMBL522748 0.74 PPARG (0.41) CYP3A4ALDH1A1KMT2AMAPTCYP1A2
SCHEMBL1529024 0.74 NR4A1 (0.38) GAANR4A1ALDH1A1MEN1KMT2A
SCHEMBL177406 0.74 MCL1 (0.49) TP53GAAALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL20641579 0.72 ALDH1A1 (0.53) TSHRTP53CA12CA1CA2
SCHEMBL14484639 0.71 ALDH1A1 (0.45) TP53CA12CA1CA2CA7
SCHEMBL17181780 0.71 ALDH1A1 (0.68) TSHRCA12CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7645773-B2 Thiazoles as inhibitors of 11β-hydroxysteroid dehydrogenase HOFFMANN-LA ROCHE INC. (US) 2010-01-12 US disclosed