SCHEMBL522748

SCHEMBL522748

Fc1cc(OBOc2ccc(Cl)c(F)c2)ccc1Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.41
PPARA Q07869 1/20 0.41
SLC6A4 P31645 6/20 0.40
HTR2A P28223 3/20 0.40
KCNH2 Q12809 3/20 0.40
GPR84 Q9NQS5 1/20 0.38
CHRNA3 P32297 1/20 0.37
ATF4 P18848 4/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
SLC6A2 P23975 2/20 0.33
SLC6A3 Q01959 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12885399 0.83 PPARG (0.42) PPARGPPARASLC6A4HTR2AKCNH2
SCHEMBL522666 0.83 SOS1 (0.46) SLC6A4HTR2AKCNH2ALDH1A1MAPT
SCHEMBL177501 0.79 HSP90AA1 (0.47) PPARGPPARASLC6A4HTR2AKCNH2
SCHEMBL177743 0.79 SOS1 (0.41) SLC6A4HTR2A
SCHEMBL1047926 0.76 PPARG (0.41) PPARGPPARASLC6A4HTR2AKCNH2
SCHEMBL276095 0.76 CYP1A2 (0.46) PPARGPPARASLC6A4HTR2AKCNH2
SCHEMBL29590981 0.76 CYP1A2 (0.46) PPARGPPARASLC6A4HTR2AKCNH2
SCHEMBL423469 0.74 ESR1 (0.41) CYP3A4
SCHEMBL3540409 0.74 TSHR (0.48) CYP1A2CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL1198940 0.74 SLC6A4 (0.38) SLC6A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250333383-A1 N-OXIDE COMPOUNDS AND USE THEREOF SK BIOPHARMACEUTICALS CO., LTD. (KR) 2025-10-30 US disclosed
EP-4514777-A1 N-OXIDE COMPOUNDS AND USE THEREOF SK Biopharmaceuticals Co., Ltd. (KR) 2025-03-05 EP disclosed
CN-117500496-A Pyrimidine and pyridinamine compounds and their use in the treatment of diseases 艾匹根生物技术有限公司 2024-02-02 CN disclosed
WO-2023211195-A1 N-OXIDE COMPOUNDS AND USE THEREOF SK BIOPHARMACEUTICALS CO., LTD. (KR) 2023-11-02 WO disclosed
US-20220363640-A1 ANTIVIRAL COMPOUNDS Janssen Biopharma, Inc. (US) 2022-11-17 US disclosed
US-20210403467-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2021-12-30 US disclosed
US-11021444-B2 Antiviral compounds Janssen Biopharma, Inc. (US) 2021-06-01 US disclosed
US-20200331907-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES ABBVIE INC (US) 2020-10-22 US disclosed
US-20190263754-A1 ANTIVIRAL COMPOUNDS ALIOS BIOPHARMA, INC. (US) 2019-08-29 US disclosed
EP-3415514-A1 APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES AbbVie Inc. (US) 2018-12-19 EP disclosed
WO-2010067069-A1 COMPOUNDS FOR USE IN THE TREATMENT OF PAIN THE UNIVERSITY OF LIVERPOOL (GB) 2010-06-17 WO disclosed
US-20080312271-A1 AZABENZIMIDAZOLYL COMPOUNDS PFIZER INC. 2008-12-18 US disclosed
US-20080280933-A1 BENZIMIDAZOLYL COMPOUNDS EFREMOV IVAN 2008-11-13 US disclosed
EP-1981876-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS Arrow Therapeutics Limited (GB) 2008-10-22 EP disclosed
WO-2008012623-A1 BENZIMIDAZOLYL COMPOUNDS AS POTENTIATORS OF MGLUR2 SUBTYPE OF GLUTAMATE RECEPTOR PFIZER PRODUCTS INC. (US) 2008-01-31 WO disclosed
WO-2008012622-A2 AZABENZIMIDAZOLYL COMPOUNDS AS POTENTIATORS OF MGLUR2 SUBTYPE OF GLUTAMATE RECEPTOR PFIZER PRODUCTS INC. (US) 2008-01-31 WO disclosed
WO-2007080401-A1 TRIAZOLOANILINOPYRIMIDINE DERIVATIVES FOR USE AS ANTIVIRAL AGENTS ARROW THERAPEUTICS LIMITED (GB) 2007-07-19 WO disclosed
EP-0456793-B1 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK PATENT GMBH (DE) 1996-10-23 EP disclosed
WO-1991009016-A2 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK PATENT GMBH (DE) 1991-06-27 WO disclosed
WO-1991009016-A1 HALOPHENYL SUBSTITUTED HETEROCYCLIC DERIVATIVES MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1991-06-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190263754-A1 ANTIVIRAL COMPOUNDS MAVS, SARS1, ZC3HAV1 PPARG 2526/4885PPARA 2015/4885SLC6A4 3882/4885
US-20250333383-A1 N-OXIDE COMPOUNDS AND USE THEREOF SCNN1B, SCN1B, SCN2B PPARG 2152/4885PPARA 2527/4885SLC6A4 146/4885
US-20080280933-A1 BENZIMIDAZOLYL COMPOUNDS PAICS, TMBIM6, ABCG2 PPARG 102/4885PPARA 513/4885SLC6A4 642/4885
US-11021444-B2 Antiviral compounds MAVS, SARS1, ZC3HAV1 PPARG 2526/4885PPARA 2015/4885SLC6A4 3882/4885
US-20220363640-A1 ANTIVIRAL COMPOUNDS MAVS, SARS1, ZC3HAV1 PPARG 2526/4885PPARA 2015/4885SLC6A4 3882/4885
US-20080312271-A1 AZABENZIMIDAZOLYL COMPOUNDS AZI2, PAICS, UGT2B7 PPARG 377/4885PPARA 1667/4885SLC6A4 719/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.