SCHEMBL3550335

SCHEMBL3550335

Cc1ccc(Cl)c(-c2ccc(C(O)C3=CCCCC3=O)cn2)c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.44
ALDH1A1 P00352 1/20 0.39
DHODH Q02127 2/20 0.33
HIF1A Q16665 1/20 0.33
MAPT P10636 1/20 0.32
TP53 P04637 1/20 0.32
ALKBH3 Q96Q83 1/20 0.32
CYP3A4 P08684 1/20 0.31
ALOX15 P16050 1/20 0.31
KDM1A O60341 1/20 0.31
PTGES O14684 1/20 0.31
CYP2C19 P33261 1/20 0.30
SMO Q99835 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855535 0.95 ALDH1A1 (0.44) THRBALDH1A1DHODHALKBH3KDM1A
SCHEMBL14400222 0.71 THRB (0.65) THRBALDH1A1HIF1AMAPTTP53
SCHEMBL2849018 0.70 THRB (0.42) THRBALDH1A1HIF1AMAPTTP53
SCHEMBL2853820 0.70 DHODH (0.39) DHODHMAPTKDM1APTGES
SCHEMBL9901550 0.69 CCR1 (0.56) DHODHTP53CYP3A4KDM1APTGES
SCHEMBL2851270 0.66 CASP1 (0.47) ALDH1A1DHODHMAPTTP53CYP3A4
SCHEMBL5792543 0.65 THRB (0.64) THRBALDH1A1HIF1AMAPTTP53
SCHEMBL439072 0.64 KDM4E (0.43) DHODHHIF1ATP53CYP3A4KDM1A
SCHEMBL2849068 0.63 THRB (0.40) THRBALDH1A1HIF1AMAPTTP53
SCHEMBL2850977 0.62 ALDH1A1 (0.41) THRBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7666883-B2 2-[(2-Chloro-5-methyl pyridine-3-yl)(hydroxy)methyl]acrylonitrile; against chloroquine sensitive and chloroquine resistant Plasmodium falciparum; treating malarial; chemical preparation COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2010-02-23 US disclosed
US-20070117822-A1 Novel antimalarial baylis-hillman adducts and a process for the preparation thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2007-05-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070117822-A1 Novel antimalarial baylis-hillman adducts and a process for the preparation thereof HBS1L, SSBP1, QARS1 THRB 4830/4885ALDH1A1 1459/4885DHODH 49/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.