SCHEMBL3551983

SCHEMBL3551983

O=C(O)c1ccc(C(Cl)(Cl)c2ccc(C(=O)O)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.60
TP53 P04637 1/20 0.60
ALOX15 P16050 1/20 0.54
SRD5A2 P31213 6/20 0.54
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
CA12 O43570 1/20 0.50
CA3 P07451 1/20 0.50
TYR P14679 1/20 0.50
DRD1 P21728 1/20 0.50
CA4 P22748 1/20 0.50
CA6 P23280 1/20 0.50
CA5A P35218 1/20 0.50
CA7 P43166 1/20 0.50
CA9 Q16790 1/20 0.50
CA14 Q9ULX7 1/20 0.50
CA5B Q9Y2D0 1/20 0.50
RARB P10826 1/20 0.48
RARG P13631 1/20 0.48
TPMT P51580 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL365481 0.93 TSHR (0.54) TSHRTP53ALOX15SRD5A2CA1
SCHEMBL3370870 0.85 TSHR (0.60) TSHRTP53ALOX15SRD5A2CA1
Methane SCHEMBL11452166 0.83 TSHR (0.57) TSHRTP53ALOX15SRD5A2CA1
Chloromethane SCHEMBL11451992 0.83 SRD5A2 (0.57) TSHRTP53ALOX15SRD5A2CA1
Hydrochloric Acid SCHEMBL11249823 0.83 TSHR (0.57) TSHRTP53ALOX15SRD5A2CA1
Terephthalic Acid SCHEMBL1243625 0.81 TSHR (0.80) TSHRTP53ALOX15SRD5A2CA1
SCHEMBL10915980 0.80 ALDH1A1 (0.45) TSHRTP53ALOX15SRD5A2ALDH1A1
SCHEMBL931931 0.79 TSHR (0.54) TSHRTP53ALOX15SRD5A2CA1
Terephthalic Acid SCHEMBL23302228 0.79 TSHR (0.67) TSHRTP53ALOX15SRD5A2CA1
Terephthalic Acid SCHEMBL31286876 0.79 TSHR (0.67) TSHRTP53ALOX15SRD5A2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1763560-B1 POLYARYLATE COMPOSITIONS SABIC INNOVATIVE PLASTICS IP (NL) 2009-08-26 EP claimed
EP-1763560-A1 POLYARYLATE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2007-03-21 EP claimed
US-7109274-B2 Polyarylate compositions GENERAL ELECTRIC COMPANY (US) 2006-09-19 US claimed
WO-2006012161-A1 POLYARYLATE COMPOSITIONS GENERAL ELECTRIC COMPANY (US) 2006-02-02 WO claimed
US-20060004152-A1 Polyarylate compositions GENERAL ELECTRIC COMPANY 2006-01-05 US claimed
EP-1945696-B1 METHOD OF IMPROVING ABRASION RESISTANCE OF PLASTIC ARTICLE USING FUNCTIONALIZED POLYMERS AND ARTICLE PRODUCED THEREBY SABIC INNOVATIVE PLASTICS IP (NL) 2013-07-31 EP disclosed
US-7855241-B2 Method of improving abrasion resistance of plastic article using nanoparticles and article produced thereby SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2010-12-21 US disclosed
EP-1763560-B1 POLYARYLATE COMPOSITIONS SABIC INNOVATIVE PLASTICS IP (NL) 2009-08-26 EP disclosed
US-7576140-B2 Via thermoplastic polycarbonates, polyestercarbonates, and cyclic polysiloxanes SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2009-08-18 US disclosed
US-7557174-B2 Carboxy-terminated oligomeric polyester compositions and method for making SABIC INNOVATIVE PLASTICS IP BV (NL) 2009-07-07 US disclosed
US-7524562-B2 Method of improving abrasion resistance of plastic article using functionalized polymers and article produced thereby SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2009-04-28 US disclosed
EP-1951791-A2 METHOD OF IMPROVING ABRASION RESISTANCE OF PLASTIC ARTICLE AND ARTICLE PRODUCED THEREBY General Electric Company (US) 2008-08-06 EP disclosed
US-4256625-A PERFLUOROALKENYLOXY, N-PHOSPHATOALKYL-SULFAMOYL-BENZENE SURFACTANT HOOKER CHEMICALS & PLASTICS CORP. (US) 1981-03-17 US disclosed
US-4187259-A Polymer blends with improved hydrolytic stability comprising a linear aromatic polyester and a methacrylate cross-linked acrylate copolymer HOOKER CHEMICALS & PLASTICS CORP. (US) 1980-02-05 US disclosed
US-4137278-A TRANSESTERIFICATION CATALYST HOOKER CHEMICALS & PLASTICS CORP. (US) 1979-01-30 US disclosed
US-4126602-A THERMOPLASTIC, MOLDING, HYDROLYTIC STABILITY HOOKER CHEMICALS & PLASTICS CORP. (US) 1978-11-21 US disclosed
US-4079034-A AROMATIC POLYESTER OF AN AROMATIC DICARBOXYLIC ACID AND A HALOGENATED BISPHENOL HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1978-03-14 US disclosed
US-4051106-A High molecular weight copolyester resins having a high degree of alternating structure HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1977-09-27 US disclosed
US-4051107-A Microstructured high molecular weight-low viscosity polyester polymers HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1977-09-27 US disclosed
US-4049629-A PREPARING POLYESTERS BY REACTING A DIACID HALIDE AND A SUBSTITUTED BISPHENOL AND A GLYCOL HOOKER CHEMICALS & PLASTICS CORPORATION (US) 1977-09-20 US disclosed