SCHEMBL3554040

SCHEMBL3554040

OC(=S)c1cccc(C(F)(F)F)c1

nearest known ligand 0.62

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.62
SRD5A2 P31213 1/20 0.56
LMNA P02545 2/20 0.53
GAA P10253 2/20 0.50
MAOB P27338 1/20 0.50
KCNK3 O14649 1/20 0.50
NPSR1 Q6W5P4 2/20 0.49
P2RX1 P51575 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MAPT P10636 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
POLB P06746 1/20 0.47
HPGD P15428 1/20 0.47
MGLL Q99685 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11545126 0.98 CES2 (0.60) CES2SRD5A2LMNAGAAMAOB
SCHEMBL3543279 0.84 SRD5A2 (0.45) CES2SRD5A2LMNAGAAMAOB
SCHEMBL10672352 0.83 CES2 (0.62) CES2SRD5A2LMNAGAANPSR1
SCHEMBL10842400 0.83 CES2 (0.67) CES2SRD5A2LMNAMAOBKCNK3
SCHEMBL1449175 0.82 CES2 (0.60) CES2SRD5A2LMNAGAANPSR1
SCHEMBL1198420 0.82 CES2 (0.60) CES2SRD5A2GAA
SCHEMBL4086253 0.80 CES2 (0.69) CES2SRD5A2LMNAMAOBKCNK3
SCHEMBL29433907 0.79 SRD5A2 (0.77) CES2SRD5A2LMNAMAOBKCNK3
SCHEMBL40186 0.79 SRD5A2 (0.77) CES2SRD5A2LMNAMAOBKCNK3
SCHEMBL17894211 0.79 CES2 (0.62) CES2SRD5A2LMNAGAAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012075242-A2 CONTROLLED CHEMICAL RELEASE OF HYDROGEN SULFIDE WASHINGTON STATE UNIVERSITY RESEARCH FOUNDATION (US) 2012-06-07 WO disclosed
CN-1805748-B 2-aminopyrimidine derivatives as RAF kinase inhibitors NOVARTIS AG 2010-05-26 CN disclosed
US-7691843-B2 N-hydroxyamide derivatives possessing antibacterial activity PFIZER INC. (US) 2010-04-06 US disclosed
US-20080058304-A1 N-hydroxyamide derivatives possessing antibacterial activity VICURON HOLDINGS LLC 2008-03-06 US disclosed
EP-1539744-A4 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARM INC (US) 2007-06-06 EP disclosed
CN-1805748-A 2-aminopyrimidine derivatives as RAF kinase inhibitors NOVARTIS AG (CH) 2006-07-19 CN disclosed
EP-1539744-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY Vicuron Pharmaceuticals, Inc. (US) 2005-06-15 EP disclosed
WO-2004007444-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARMACEUTICALS, INC. (US) 2004-01-22 WO disclosed
EP-0167919-B1 BENZODIAZEPINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM MERCK & CO. INC. (US) 1993-05-05 EP disclosed
US-5204482-A Ethylenediamine monoamide heteroaryl derivatives HOFFMAN-LAROCHE INC. (US) 1993-04-20 US disclosed
US-5011849-A Monoamine oxidase inhibitors HOFFMANN-LA ROCHE INC. (US) 1991-04-30 US disclosed
US-5004741-A Cholecystokinin(CCK); Treating Disorders Of The Gastrointestinal Tract, Central Nervous System And Of The Appetite Of Animals MERCK & CO., INC. (US) 1991-04-02 US disclosed
US-4820834-A Benzodiazepine analogs MERCK & CO., INC. (US) 1989-04-11 US disclosed
EP-0284256-A1 Benzodiazepine analogs MERCK & CO. INC. (US) 1988-09-28 EP disclosed
EP-0167919-A2 Benzodiazepine derivatives and pharmaceutical compositions containing them MERCK & CO. INC. (US) 1986-01-15 EP disclosed
US-4296092-A Mucolytic benzene and thiophene-carbothioic acid 2-aminoalkyl ester acid salts A. H. ROBINS COMPANY, INC. (US) 1981-10-20 US disclosed
US-4198428-A PESTICIDES, MICROBIOCIDES, MOLLUSCOCIDES BAYER AKTIENGESELLSCHAFT (DE) 1980-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080058304-A1 N-hydroxyamide derivatives possessing antibacterial activity AMDHD2, OGA, ENGASE CES2 625/4885SRD5A2 2467/4885LMNA 3400/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.