SCHEMBL3565075

SCHEMBL3565075

O=C1C(=CNc2ccc([N+](=O)[O-])cc2)c2ccccc2C(=O)N1c1ccc(Cl)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN2A Q99250 3/20 0.60
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
AMY1A P0DUB6 1/20 0.43
CA12 O43570 2/20 0.40
CA9 Q16790 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
PGR P06401 3/20 0.39
MDM2 Q00987 1/20 0.39
MAPT P10636 3/20 0.38
APP P05067 2/20 0.38
SNCA P37840 2/20 0.38
AR P10275 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3565074 1.00 SCN2A (0.60) SCN2AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3576525 0.85 MEN1 (0.57) SCN2AMEN1KMT2AALDH1A1CA12
SCHEMBL3576527 0.85 MEN1 (0.57) SCN2AMEN1KMT2AALDH1A1CA12
SCHEMBL1973251 0.78 SCN2A (1.00) SCN2AMEN1KMT2AALDH1A1CA12
SCHEMBL30118348 0.78 SCN2A (1.00) SCN2AMEN1KMT2AALDH1A1CA12
SCHEMBL3575951 0.74 ALDH1A1 (0.52) SCN2AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3575950 0.74 ALDH1A1 (0.52) SCN2AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3563214 0.74 ALDH1A1 (0.62) SCN2AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3563218 0.74 ALDH1A1 (0.62) SCN2AMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL3565158 0.73 CASP3 (0.44) MEN1KMT2AALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7713994-B2 Substituted isoquinoline-1,3(2H,4H)-diones, 1-thioxo,1,4-dihydro-2H-isoquinoline-3-ones and 1,4-dihyro-3 (2H)-isoquinolones and methods of use thereof WYETH LLC (US) 2010-05-11 US claimed