SCHEMBL3569459

SCHEMBL3569459

C[C@H](N)C(=O)NCC(Cc1ccccc1)C1=COCO1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 3/20 0.43
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
MMP2 P08253 4/20 0.41
LAP3 P28838 3/20 0.39
ANPEP P15144 1/20 0.39
RNPEP Q9H4A4 1/20 0.39
DNPEP Q9ULA0 1/20 0.39
CYP3A4 P08684 1/20 0.38
TSHR P16473 1/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3562176 1.00 CTRB1 (0.43) CTRB1MTNR1AMTNR1BMMP2LAP3
SCHEMBL3559808 0.91 MTNR1A (0.41) CTRB1MTNR1AMTNR1BMMP2LAP3
SCHEMBL1011206 0.85 MTNR1A (0.60) CTRB1MTNR1AMTNR1BCYP3A4
SCHEMBL3559900 0.81 MTNR1A (0.43) MTNR1AMTNR1BMMP2CYP3A4HDAC1
SCHEMBL3559731 0.81 MTNR1A (0.42) MTNR1AMTNR1BMMP2CYP3A4
SCHEMBL4991230 0.76 L3MBTL1 (0.50) MTNR1AMTNR1B
SCHEMBL3563505 0.76 MIF (0.43) MTNR1AMTNR1B
SCHEMBL15547346 0.76 MTNR1A (0.43) CTRB1MTNR1AMTNR1BCYP3A4
SCHEMBL1430902 0.76 MIF (0.56) MTNR1AMTNR1B
SCHEMBL5884516 0.76 MTNR1A (0.41) MTNR1AMTNR1BCYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7825256-B2 Inducible nitric oxide synthase dimerization inhibitors KALYPSYS, INC. (US) 2010-11-02 US disclosed
EP-1817030-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS Kalypsys, Inc. (US) 2007-08-15 EP disclosed
WO-2006060424-A2 INDUCIBLE NITRIC OXIDE SYNTHASE DIMERIZATION INHIBITORS KALYPSYS, INC. (US) 2006-06-08 WO disclosed