Choline

Choline

SCHEMBL357235

C[N+](C)(C)CCO.O=S(=O)([O-])C(F)(F)C(F)F

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADORA1ADORA2AADORA2BADORA3GNRHRMPLPDE3APDE3BPDE4APDE4BPDE4CPDE4DPPARASLC5A2

The experimentally established mechanism targets of Choline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
KMT2A Q03164 1/20 0.41
CYP3A4 P08684 1/20 0.41
SLC5A7 Q9GZV3 1/20 0.41
BBOX1 O75936 1/20 0.34
APAF1 O14727 1/20 0.32
POLB P06746 1/20 0.32
GRK2 P25098 1/20 0.32
DNMT1 P26358 1/20 0.32
PTPN7 P35236 1/20 0.32
RECQL P46063 1/20 0.32
BLM P54132 1/20 0.32
PPP1CA P62136 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
PTPN22 Q9Y2R2 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358111 0.85
Choline SCHEMBL27857086 0.84 MEN1 (0.43) MEN1LMNAKMT2ACYP3A4SLC5A7
Trifluoromethanesulfonic Acid SCHEMBL3785097 0.83 MEN1 (0.50) MEN1LMNAKMT2ACYP3A4SLC5A7
SCHEMBL16107569 0.81 BBOX1 (0.41) MEN1LMNAKMT2ABBOX1APAF1
Choline SCHEMBL339062 0.76 MEN1 (0.63) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL2351951 0.76 MEN1 (0.63) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL339064 0.74 MEN1 (0.60) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL3790708 0.74 MEN1 (0.60) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL3790706 0.74 MEN1 (0.60) MEN1LMNAKMT2ACYP3A4SLC5A7
Choline SCHEMBL872580 0.74 MEN1 (0.60) MEN1LMNAKMT2ACYP3A4SLC5A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414476-A1 IONIC COMPOUNDS IN LITHIUM BROMIDE/WATER ABSORPTION CYCLE SYSTEMS E. I. du Pont de Nemours and Company (US) 2012-02-08 EP claimed
WO-2010117836-A1 IONIC COMPOUNDS IN LITHIUM BROMIDE/WATER ABSORPTION CYCLE SYSTEMS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-10-14 WO claimed
EP-2414476-A1 IONIC COMPOUNDS IN LITHIUM BROMIDE/WATER ABSORPTION CYCLE SYSTEMS E. I. du Pont de Nemours and Company (US) 2012-02-08 EP disclosed
US-20120011886-A1 IONIC COMPOUNDS IN LITHIUM BROMIDE/WATER ABSORPTION CYCLE SYSTEMS E. I. DU PONT DE NEMOURS AND COMPANY 2012-01-19 US disclosed
WO-2010117836-A1 IONIC COMPOUNDS IN LITHIUM BROMIDE/WATER ABSORPTION CYCLE SYSTEMS E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-10-14 WO disclosed