SCHEMBL357502

SCHEMBL357502

C=C(C)C(Cc1ccccc1)(OC(N)=O)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.40
HIF1A Q16665 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRD1 P41143 2/20 0.39
TSHR P16473 2/20 0.37
TRPA1 O75762 1/20 0.37
KCNH2 Q12809 2/20 0.37
MRGPRX2 Q96LB1 1/20 0.37
CHRM3 P20309 1/20 0.37
HRH2 P25021 1/20 0.37
HTR2A P28223 1/20 0.37
ADRA1A P35348 1/20 0.37
OPRK1 P41145 1/20 0.37
ALDH1A1 P00352 3/20 0.37
RECQL P46063 1/20 0.37
MAPK1 P28482 1/20 0.37
ALPI P09923 1/20 0.37
PKM P14618 1/20 0.37
PTGS1 P23219 1/20 0.37
XIAP P98170 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2641207 0.79 PPARG (0.44) SMN1; SMN2HIF1AALDH1A1RECQLMAPK1
SCHEMBL9049038 0.75 TRPA1 (0.45) SMN1; SMN2HIF1AOPRM1OPRD1TSHR
SCHEMBL3656311 0.73 SMN1; SMN2 (0.48) SMN1; SMN2HIF1ATRPA1ALDH1A1RECQL
SCHEMBL9278784 0.73 HIF1A (0.48) SMN1; SMN2HIF1ATRPA1ALDH1A1RECQL
SCHEMBL6837561 0.71 PPARG (0.49) SMN1; SMN2HIF1AOPRM1OPRD1TSHR
SCHEMBL27768873 0.69 SMN1; SMN2 (0.48) SMN1; SMN2HIF1AOPRM1OPRD1TSHR
SCHEMBL1547275 0.69 HIF1A (0.44) SMN1; SMN2HIF1ATSHRTRPA1ALDH1A1
SCHEMBL7619909 0.69 SLC6A2 (0.48) SMN1; SMN2HIF1AOPRM1OPRD1KCNH2
SCHEMBL6461316 0.69 SMN1; SMN2 (0.44) SMN1; SMN2HIF1ATSHRALDH1A1RECQL
SCHEMBL412308 0.68 SMN1; SMN2 (0.52) SMN1; SMN2HIF1AOPRM1OPRD1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 253 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2104715-B1 METHOD FOR PRODUCING A WATER SELF DISPERSIBLE METALLIC OXIDE AND HYDROXIDE POWDER, POWDER AND USES THEREOF COATEX SAS (FR) 2019-03-20 EP claimed
EP-2976392-B1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX SAS (FR) 2018-04-25 EP claimed
EP-2222920-B1 METHOD FOR MANUFACTURING A COATING SLIP INCLUDING THE USE OF AN ACRYLIC THICKENER WITH A WATER RESISTANT CHAIN AND SLIP OBTAINED OMYA INT AG (CH) 2018-02-07 EP claimed
EP-2108007-B1 USE OF A RHEOLOGIC ADDITIVE IN THE VIBRO-COMPACTION PRODUCTION OF A FORMULATION CONTAINING WATER AND A HYDRAULIC BINDER, AND FORMULATION THUS OBTAINED COATEX SAS (FR) 2016-04-13 EP claimed
EP-2976392-A1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX (FR) 2016-01-27 EP claimed
EP-2129468-B1 USE AS RHEOLOGICAL AGENT IN CHARGED PLASTIC PASTE, OF DRY-GROUND CALCIUM CARBONATE WITH (METH)ACRYLIC ACID COPOLYMER WITH ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION COATEX SAS (FR) 2015-12-09 EP claimed
WO-2014147321-A1 USE OF A POLYMERIC EMULSION FOR THE SURFACE TREATMENT OF THE PARTICLES OF AN INORGANIC MATERIAL COATEX (FR) 2014-09-25 WO claimed
US-8637579-B2 Process to thicken aqueous compositions by means of organophosphate polymers COATEX S.A.S. (FR) 2014-01-28 US claimed
EP-2125235-B1 USE IN HYDRAULIC BINDER COMPOSITION OF DRY-GROUND CALCIUM CARBONATE WITH (METH)ACRYLIC ACID COPOLYMER AND ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION COATEX SAS (FR) 2013-11-27 EP claimed
EP-2379649-B1 PROCESS TO PREPARE SELF-BINDING PIGMENT PARTICLES IMPLEMENTING ACRYLIC COMB COPOLYMERS WITH HYDROPHOBIC GROUPS AS COUPLING AGENTS, SELF BINDING PIGMENT PARTICLES AND USES THEREOF OMYA INT AG (CH) 2013-11-13 EP claimed
EP-1708803-A2 USE OF STRUCTURED WATER-SOLUBLE POLYMERS OBTAINED BY CONTROLLED RADICAL POLYMERIZATION AS A DISPERSANT AND AGENT FOR ASSISTING IN THE GRINDING OF MINERAL MATERIALS COATEX S.A.S. (FR) 2006-10-11 EP claimed
US-20060162884-A1 Novel inorganic pigment containing calcium carbonate, aqueous suspension containing same, and uses thereof OMYA INTERNATIONAL AG (CH) 2006-07-27 US claimed
US-20060142498-A1 gloss activator for sheet of paper, irrespective of viewing angle; paper coating; weakly ionic water soluble acrylic-polyether (or silyloxyether) graft addition-condensation copolymer OMYA INTERNATIONAL AG (CH) 2006-06-29 US claimed
WO-2006048539-A1 SUBSTITUTED CUMYL PHENOLS, USE THEREOF IN A COPOLYMERISATION METHOD COPOLYMERS THUS OBTAINED AND USE THEREOF AS THICKENERS COATEX S.A.S. (FR) 2006-05-11 WO claimed
US-20060009560-A1 Aqueous suspensions of ground mineral materials, with low ion load and their uses OMYA INTERNATIONAL AG (CH) 2006-01-12 US claimed
EP-1572764-A1 AQUEOUS SUSPENSIONS OF GROUND MINERAL MATERIALS, WITH LOW ION LOAD AND THEIR USES Omya AG (CH) 2005-09-14 EP claimed
EP-1565504-A1 USE OF A COPOLYMER HAVING AT LEAST ONE GRAFTED ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION AS AN AGENT FOR IMPROVING OPTICAL BRIGHTENING ACTIVATION, AND PRODUCTS OBTAINED COATEX S.A.S. (FR) 2005-08-24 EP claimed
WO-2005063371-A2 USE OF STRUCTURED WATER-SOLUBLE POLYMERS OBTAINED BY CONTROLLED RADICAL POLYMERIZATION AS A DISPERSANT AND AGENT FOR ASSISTING IN THE GRINDING OF MINERAL MATERIALS COATEX S.A.S. (FR) 2005-07-14 WO claimed
WO-2004044022-A1 USE OF A COPOLYMER HAVING AT LEAST ONE GRAFTED ALKOXY OR HYDROXY POLYALKYLENE GLYCOL FUNCTION AS AN AGENT FOR IMPROVING OPTICAL BRIGHTENING ACTIVATION, AND PRODUCTS OBTAINED COATEX S.A.S. (FR) 2004-05-27 WO claimed
WO-2004041882-A1 AQUEOUS SUSPENSIONS OF GROUND MINERAL MATERIALS, WITH LOW ION LOAD AND THEIR USES OMYA AG (CH) 2004-05-21 WO claimed