SCHEMBL3580139

SCHEMBL3580139

NCc1ccn(-c2cccc(-c3nc4cccc(C(N)=O)c4[nH]3)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.46
KDR P35968 1/20 0.46
PARP1 P09874 18/20 0.41
PIM1 P11309 1/20 0.36
PIM3 Q86V86 1/20 0.36
DHODH Q02127 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582143 0.90 AURKB (0.56) AURKBKDRPARP1DHODH
SCHEMBL3586255 0.85 KDR (0.41) AURKBKDRPARP1CYP3A4CYP2C9
SCHEMBL3576439 0.84 KDR (0.38) AURKBKDRPARP1DHODHCYP3A4
SCHEMBL3580135 0.84 AURKB (0.61) AURKBKDRPARP1PIM1PIM3
SCHEMBL3584745 0.81 PARP1 (0.39) AURKBPARP1PIM1PIM3DHODH
SCHEMBL3580644 0.77 AURKB (0.76) AURKBKDRPARP1DHODH
SCHEMBL7136552 0.76 PARP1 (0.52) AURKBPARP1PIM1PIM3DHODH
SCHEMBL3578629 0.76 AURKB (0.64) AURKBKDRPARP1DHODH
SCHEMBL3582340 0.76 AURKB (0.63) AURKBKDRPARP1PIM1PIM3
SCHEMBL6807111 0.75 PARP1 (0.46) AURKBKDRPARP1PIM1PIM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed