SCHEMBL3584745

SCHEMBL3584745

NCc1cccn1-c1cccc(-c2nc3cccc(C(N)=O)c3[nH]2)c1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.39
PIM1 P11309 2/20 0.36
PIM3 Q86V86 2/20 0.36
AURKB Q96GD4 2/20 0.36
DYRK3 O43781 1/20 0.36
MAP4K4 O95819 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CSNK2A1 P68400 1/20 0.36
PKN2 Q16513 1/20 0.36
BRSK1 Q8TDC3 1/20 0.36
HIPK2 Q9H2X6 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
MKNK2 Q9HBH9 1/20 0.36
STK17A Q9UEE5 1/20 0.36
MAP4K5 Q9Y4K4 1/20 0.36
DHODH Q02127 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
BTK Q06187 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3584741 0.84 PARP1 (0.59) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL3580139 0.81 AURKB (0.46) PARP1PIM1PIM3AURKBDHODH
SCHEMBL3582864 0.76 GRK6 (0.48) PARP1CYP3A4CYP2C9
SCHEMBL3585144 0.75 PARP1 (0.64) PARP1PIM1AURKBMAP4K4HIPK2
SCHEMBL7136552 0.75 PARP1 (0.52) PARP1PIM1PIM3AURKBDHODH
SCHEMBL3576439 0.75 KDR (0.38) PARP1AURKBPKN2DHODHCYP3A4
SCHEMBL3579908 0.75 PARP1 (0.61) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL3580302 0.74 DYRK3 (0.54) PARP1PIM1PIM3AURKBDYRK3
SCHEMBL29696369 0.74 NPC1 (0.53) PARP1DHODHCYP3A4CYP2C9
SCHEMBL3575207 0.74 DYRK3 (0.53) PARP1PIM1PIM3AURKBDYRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed