SCHEMBL3586255

SCHEMBL3586255

NC(=O)c1cccc2nc(-c3cccc(-n4ccc(CNC(=O)C(F)(F)F)c4)c3)[nH]c12

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.41
AURKB Q96GD4 1/20 0.41
PARP1 P09874 17/20 0.37
ELANE P08246 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
KCNH2 Q12809 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3582780 0.91 AURKB (0.49) KDRAURKBPARP1ELANEKCNH2
SCHEMBL3586249 0.86 KDR (0.54) KDRAURKBPARP1
SCHEMBL3580139 0.85 AURKB (0.46) KDRAURKBPARP1CYP3A4CYP2C9
SCHEMBL6582952 0.78 KDR (0.41) KDRAURKBPARP1
SCHEMBL3577370 0.78 KDR (0.65) KDRAURKBPARP1
SCHEMBL3576439 0.77 KDR (0.38) KDRAURKBPARP1CYP3A4CYP2C9
SCHEMBL3582143 0.75 AURKB (0.56) KDRAURKBPARP1
SCHEMBL3580644 0.71 AURKB (0.76) KDRAURKBPARP1
SCHEMBL3584745 0.71 PARP1 (0.39) AURKBPARP1CYP3A4CYP2C9
SCHEMBL3578629 0.70 AURKB (0.64) KDRAURKBPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed