SCHEMBL3580975

SCHEMBL3580975

CN(C#N)c1ccc(Cl)c(Cl)c1C(=O)N(CCc1cccc(C(F)(F)F)c1)Cc1ccc(C2CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.34
GRK5 P34947 1/20 0.34
CDK8 P49336 1/20 0.34
S1PR5 Q9H228 1/20 0.34
PGR P06401 1/20 0.34
KCNH2 Q12809 1/20 0.34
SLC2A1 P11166 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
ATM Q13315 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
STAT3 P40763 1/20 0.33
CCR1 P32246 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27730389 0.92 S1PR1 (0.37) S1PR1GRK5CDK8S1PR5PGR
SCHEMBL3586256 0.89 STAT3 (0.35) KCNH2STAT3
SCHEMBL3580976 0.87 MCL1 (0.35) S1PR1GRK5CDK8S1PR5PGR
SCHEMBL27730380 0.87 LMNA (0.34) S1PR1GRK5CDK8S1PR5PGR
SCHEMBL3577794 0.87 LMNA (0.37) S1PR1GRK5CDK8S1PR5KCNH2
SCHEMBL3578656 0.84 MCL1 (0.37) S1PR1GRK5CDK8S1PR5SLC2A1
SCHEMBL3581173 0.84 CCR1 (0.37) S1PR1GRK5CDK8S1PR5KCNH2
SCHEMBL3579273 0.83 LMNA (0.37) S1PR1GRK5CDK8S1PR5MEN1
SCHEMBL27730387 0.82 S1PR1 (0.36) S1PR1GRK5CDK8S1PR5PGR
SCHEMBL27730488 0.81 SLC6A9 (0.35) KCNH2STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7678818-B2 Anthranilamide and 2-amino-heteroarene-carboxamide compounds HOFFMANN-LA ROCHE INC. (US) 2010-03-16 US claimed
EP-1984340-B1 ANTHRANILAMIDE/2-AMINO-HETEROARENE CARBOXAMIDE DERIVATIVES HOFFMANN LA ROCHE (CH) 2012-06-27 EP disclosed