SCHEMBL3582857

SCHEMBL3582857

NC(=O)c1cccc2[nH]c(-c3cccc(N4CCNCC4)c3)nc12

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 18/20 0.66
DHODH Q02127 1/20 0.59
PARP2 Q9UGN5 1/20 0.58
PKN1 Q16512 2/20 0.56
PKN2 Q16513 2/20 0.56
PLK4 O00444 1/20 0.56
MAPK13 O15264 1/20 0.56
DYRK3 O43781 1/20 0.56
ROCK2 O75116 1/20 0.56
RPS6KA5 O75582 1/20 0.56
PRKD3 O94806 1/20 0.56
MAP4K4 O95819 1/20 0.56
CHEK2 O96017 1/20 0.56
PIM1 P11309 1/20 0.56
PHKG2 P15735 1/20 0.56
PRKACA P17612 1/20 0.56
RPS6KB1 P23443 1/20 0.56
CSNK1D P48730 1/20 0.56
CLK2 P49760 1/20 0.56
GSK3A P49840 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580352 0.89 AURKB (0.68) PARP1DHODHPARP2PKN1PKN2
SCHEMBL3582368 0.85 AURKB (0.64) PARP1DHODHPARP2PKN1PKN2
SCHEMBL6580875 0.84 PARP1 (0.48) PARP1MKNK2
SCHEMBL3584970 0.83 PARP1 (0.53) PARP1PARP2DYRK3PRKD3MAP4K4
SCHEMBL31413225 0.83 PARP1 (0.66) PARP1DHODH
SCHEMBL3582864 0.83 GRK6 (0.48) PARP1CHEK2
SCHEMBL6805718 0.81 AURKA (0.72) PARP1DHODHPARP2PKN1PKN2
SCHEMBL3585138 0.80 PARP1 (1.00) PARP1DHODHPARP2PKN1PKN2
SCHEMBL5621808 0.79 PARP1 (0.72) PARP1PARP2
SCHEMBL31413270 0.78 PARP1 (0.82) PARP1DHODHPARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed