SCHEMBL3582373

SCHEMBL3582373

NC(=O)c1cccc2nc(-c3ccc(N4CCCNCC4)cc3)[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.49
AURKA O14965 1/20 0.47
AURKB Q96GD4 1/20 0.47
CHEK2 O96017 6/20 0.46
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
ATR Q13535 3/20 0.42
PARP2 Q9UGN5 2/20 0.42
PIM1 P11309 1/20 0.41
PIM3 Q86V86 1/20 0.41
PIM2 Q9P1W9 1/20 0.41
ACVR1 Q04771 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580358 0.96 PARP1 (0.53) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL6812407 0.86 AURKA (0.50) PARP1AURKAAURKB
SCHEMBL3582864 0.85 GRK6 (0.48) PARP1CHEK2
SCHEMBL3577227 0.84 AURKA (0.53) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3587289 0.84 AURKA (0.56) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3582368 0.83 AURKB (0.64) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL5621910 0.82 HTR3A (0.48) PARP1CHRNB2CHRNA4PIM1
SCHEMBL3579920 0.82 AURKA (0.49) PARP1AURKAAURKBCHEK2PARP2
SCHEMBL3582849 0.82 AURKB (0.58) PARP1AURKAAURKBCHEK2
SCHEMBL3584976 0.82 ACVR1 (0.42) PARP1AURKAAURKBCHEK2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed