SCHEMBL358333

SCHEMBL358333

CC(=O)N1CCC(n2nc3c(C(N)=O)cccc3c2-c2ccccc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.48
MAP3K7 O43318 2/20 0.40
TAB1 Q15750 2/20 0.40
ACACB O00763 3/20 0.40
ACACA Q13085 3/20 0.40
SMO Q99835 1/20 0.39
BTK Q06187 1/20 0.39
CNR1 P21554 1/20 0.38
BRD4 O60885 1/20 0.38
RPS6KB1 P23443 2/20 0.38
AURKA O14965 2/20 0.38
NCF1 P14598 1/20 0.38
AURKB Q96GD4 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
TP53 P04637 1/20 0.38
ALOX15 P16050 1/20 0.38
MAPK1 P28482 1/20 0.38
CASP1 P29466 1/20 0.38
CASP7 P55210 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL358330 0.89 PARP1 (0.47) PARP1CNR1RPS6KB1AURKAAURKB
SCHEMBL10172648 0.88 PARP1 (0.41) PARP1BTKCNR1RPS6KB1AURKA
SCHEMBL359223 0.86 PARP1 (0.49) PARP1BTK
SCHEMBL10173016 0.85 PARP1 (0.51) PARP1MAP3K7TAB1ACACBACACA
Hydrochloric Acid SCHEMBL357948 0.82 RPS6KB1 (0.48) PARP1RPS6KB1AURKAPARP2
SCHEMBL370739 0.81 PARP1 (0.46) PARP1
SCHEMBL27917093 0.80 PIK3CA (0.39) ACACBACACASMOBTKCNR1
SCHEMBL370599 0.78 PARP1 (0.46) PARP1
SCHEMBL368905 0.77 PARP1 (0.49) PARP1
SCHEMBL358670 0.72 PARP1 (0.52) PARP1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO claimed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed