SCHEMBL358330

SCHEMBL358330

CN1CCC(n2nc3c(C(N)=O)cccc3c2-c2ccccc2)CC1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.47
PARP2 Q9UGN5 5/20 0.46
CCNA2 P20248 1/20 0.42
CDK2 P24941 1/20 0.42
CCNA1 P78396 1/20 0.42
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
KMT2A Q03164 1/20 0.40
CNR1 P21554 1/20 0.39
RPS6KB1 P23443 4/20 0.39
AURKA O14965 3/20 0.39
AURKB Q96GD4 1/20 0.39
ACVR1 Q04771 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10172648 0.90 PARP1 (0.41) PARP1PARP2KMT2ACNR1RPS6KB1
SCHEMBL358333 0.89 PARP1 (0.48) PARP1PARP2CCNA2CDK2CCNA1
Hydrochloric Acid SCHEMBL357948 0.84 RPS6KB1 (0.48) PARP1PARP2RPS6KB1AURKA
SCHEMBL359223 0.84 PARP1 (0.49) PARP1
SCHEMBL370739 0.79 PARP1 (0.46) PARP1KMT2A
SCHEMBL27899434 0.76 ADRA1A (0.37) CCNA2CDK2CCNA1KMT2ACNR1
SCHEMBL370599 0.76 PARP1 (0.46) PARP1
SCHEMBL10173016 0.74 PARP1 (0.51) PARP1PARP2KMT2ARPS6KB1AURKA
SCHEMBL359581 0.71 RPS6KB1 (0.48) PARP1PARP2RPS6KB1AURKA
SCHEMBL358670 0.69 PARP1 (0.52) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO claimed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed