SCHEMBL3584709

SCHEMBL3584709

NC(=O)c1cccc2[nH]c(-c3ccc(N4CCN(C5CCCCC5)CC4)cc3)nc12

nearest known ligand 0.64

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.64
AURKB Q96GD4 1/20 0.64
PARP1 P09874 19/20 0.61
PARP2 Q9UGN5 7/20 0.60
DHODH Q02127 2/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3589348 0.92 PARP1 (0.62) AURKAAURKBPARP1PARP2DHODH
SCHEMBL6581404 0.86 AURKB (0.47) AURKAAURKBPARP1PARP2DHODH
SCHEMBL3584716 0.84 AURKB (0.47) AURKAAURKBPARP1PARP2
SCHEMBL5620426 0.83 PARP1 (0.68) PARP1
SCHEMBL3587286 0.83 AURKA (0.76) AURKAAURKBPARP1PARP2DHODH
SCHEMBL4970545 0.83 PARP1 (0.73) PARP1PARP2
SCHEMBL7763627 0.83 GAA (0.51) AURKAAURKBPARP1
SCHEMBL3580352 0.82 AURKB (0.68) AURKAAURKBPARP1PARP2DHODH
SCHEMBL3577220 0.82 AURKA (0.71) AURKAAURKBPARP1PARP2DHODH
SCHEMBL4974007 0.82 PARP1 (0.74) PARP1PARP2DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed