SCHEMBL3584716

SCHEMBL3584716

NC(=O)c1cccc2nc(-c3ccc(N4CCN(C5CCCCC5)CC4)cc3)[nH]c12

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 2/20 0.47
AURKA O14965 1/20 0.47
PARP1 P09874 10/20 0.46
CHEK2 O96017 7/20 0.46
PARP2 Q9UGN5 2/20 0.42
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3527499 0.92 AURKB (0.45) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL3584709 0.84 AURKA (0.64) AURKBAURKAPARP1PARP2
SCHEMBL5620431 0.83 PARP1 (0.51) PARP1PARP2
SCHEMBL3587289 0.83 AURKA (0.56) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL3580358 0.82 PARP1 (0.53) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL3577227 0.82 AURKA (0.53) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL3576982 0.81 AURKA (0.52) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL5622215 0.81 PARP1 (0.48) PARP1PARP2
SCHEMBL3582373 0.81 PARP1 (0.49) AURKBAURKAPARP1CHEK2PARP2
SCHEMBL3582282 0.81 AURKB (0.61) AURKBAURKAPARP1CHEK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed