SCHEMBL3585484

SCHEMBL3585484

NC(=O)c1cccc2[nH]c(-c3ccc(N4CCCN(Cc5ccccc5)CC4)cc3)nc12

nearest known ligand 0.75

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 17/20 0.75
AURKB Q96GD4 3/20 0.72
AURKA O14965 2/20 0.72
KDR P35968 2/20 0.72
DHODH Q02127 4/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580117 0.96 AURKB (0.77) PARP1AURKBAURKAKDRDHODH
SCHEMBL3582843 0.88 AURKB (0.76) PARP1AURKBAURKAKDRDHODH
SCHEMBL6806434 0.88 AURKB (0.93) PARP1AURKBAURKAKDRDHODH
SCHEMBL6580774 0.87 PARP1 (0.56) PARP1AURKBAURKAKDRDHODH
SCHEMBL7137128 0.86 PARP1 (1.00) PARP1AURKBAURKAKDRDHODH
SCHEMBL7139308 0.85 PARP1 (1.00) PARP1AURKBAURKAKDRDHODH
SCHEMBL3585487 0.85 PARP1 (0.54) PARP1AURKBAURKAKDRDHODH
SCHEMBL5620780 0.85 AURKA (0.62) PARP1AURKBAURKAKDR
SCHEMBL3582845 0.85 AURKB (0.93) PARP1AURKBAURKAKDRDHODH
SCHEMBL3578622 0.85 AURKB (0.85) PARP1AURKBAURKAKDRDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed