SCHEMBL3585487

SCHEMBL3585487

NC(=O)c1cccc2nc(-c3ccc(N4CCCN(Cc5ccccc5)CC4)cc3)[nH]c12

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.54
AURKB Q96GD4 3/20 0.53
AURKA O14965 2/20 0.53
KDR P35968 2/20 0.53
CHEK2 O96017 4/20 0.48
JAK2 O60674 1/20 0.46
DHODH Q02127 1/20 0.46
ACHE P22303 1/20 0.45
KDM1A O60341 1/20 0.44
USP2 O75604 1/20 0.44
TP53 P04637 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3580122 0.96 AURKB (0.56) PARP1AURKBAURKAKDRCHEK2
SCHEMBL3582849 0.88 AURKB (0.58) PARP1AURKBAURKAKDRCHEK2
SCHEMBL6806441 0.88 AURKB (0.70) PARP1AURKBAURKAKDRCHEK2
SCHEMBL3582854 0.85 AURKB (0.70) PARP1AURKBAURKAKDRCHEK2
SCHEMBL3585484 0.85 PARP1 (0.75) PARP1AURKBAURKAKDRDHODH
SCHEMBL3578629 0.85 AURKB (0.64) PARP1AURKBAURKAKDRCHEK2
SCHEMBL5620788 0.85 AURKA (0.49) PARP1AURKBAURKAKDRUSP2
SCHEMBL3582282 0.84 AURKB (0.61) PARP1AURKBAURKAKDRCHEK2
SCHEMBL6805222 0.84 AURKA (0.75) PARP1AURKBAURKAKDRCHEK2
SCHEMBL3577227 0.83 AURKA (0.53) PARP1AURKBAURKACHEK2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7781596-B1 Substituted 2-phenylbenzimidazoles, the production thereof and their use ABBOTT LABORATORIES (US) 2010-08-24 US disclosed