SCHEMBL3585979

SCHEMBL3585979

O=C(O)N(c1ccccc1)c1nnc(Br)s1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 3/20 0.44
ALDH1A1 P00352 5/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
POLB P06746 2/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.35
MAPT P10636 1/20 0.34
MLYCD O95822 1/20 0.34
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4716184 0.87 ALDH1A1 (0.41) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL5381977 0.81 ALDH1A1 (0.48) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL1945009 0.80 NPC1 (0.50) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL1943555 0.78 NPC1 (0.40) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL4762222 0.78 CYP3A4 (0.47) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL5373150 0.78 GLS (0.45) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL3575822 0.77 MLYCD (0.43) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL19778 0.72 NPSR1 (0.70) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL20298486 0.70 NPSR1 (0.45) NPSR1ALDH1A1NPC1RAB9APOLB
SCHEMBL17601670 0.70 NPC1 (0.44) NPSR1ALDH1A1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100048543-A1 PYRIMIDINE COMPOUNDS HAVING TIES (TEK) INHIBITORY ACTIVITY ASTRAZENECA AB (SE) 2010-02-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100048543-A1 PYRIMIDINE COMPOUNDS HAVING TIES (TEK) INHIBITORY ACTIVITY TEK, TYMP, TIE1 NPSR1 1799/4885ALDH1A1 2198/4885NPC1 4705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.