SCHEMBL3590337

SCHEMBL3590337

O=C(O)c1cc(N(CCBr)CCBr)c([N+](=O)[O-])cc1[N+](=O)[O-]

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 4/20 0.47
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 2/20 0.41
DTYMK P23919 1/20 0.41
HTT P42858 2/20 0.40
TP53 P04637 1/20 0.40
GLA P06280 1/20 0.39
POLB P06746 2/20 0.36
ALDH3A1 P30838 1/20 0.36
LMNA P02545 1/20 0.36
TSHR P16473 1/20 0.36
MAPT P10636 2/20 0.35
CYP3A4 P08684 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
CASP6 P55212 1/20 0.35
GPR35 Q9HC97 1/20 0.35
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8636703 0.87 MAPT (0.50) HCAR3ALDH1A1KDM4EHTTPOLB
SCHEMBL13545666 0.85 HCAR3 (0.64) HCAR3ALDH1A1KDM4EDTYMKHTT
SCHEMBL3582922 0.85 HCAR3 (0.47) HCAR3ALDH1A1KDM4EDTYMKHTT
SCHEMBL3579835 0.83 HCAR3 (0.41) HCAR3ALDH1A1KDM4EDTYMKHTT
SCHEMBL28153049 0.83 HCAR3 (0.54) HCAR3ALDH1A1KDM4EDTYMKHTT
SCHEMBL3421496 0.82 MAPT (0.46) HCAR3ALDH1A1KDM4EPOLBALDH3A1
SCHEMBL2970718 0.81 MAPT (0.45) HCAR3ALDH1A1KDM4EPOLBALDH3A1
SCHEMBL13202973 0.81 MAPT (0.45) HCAR3ALDH1A1KDM4EPOLBALDH3A1
SCHEMBL367596 0.80 ALDH1A1 (0.41) HCAR3ALDH1A1KDM4EPOLBLMNA
SCHEMBL3983950 0.80 MAPT (0.46) HCAR3ALDH1A1KDM4EHTTGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100010094-A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents AUCKLAND UNISERVICES LIMITED (NZ) 2010-01-14 US disclosed
US-7629332-B2 Nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents AUCKLAND UNISERVICES LIMITED (NZ) 2009-12-08 US disclosed
US-20070032455-A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents AUCKLAND UNIVERVICES LIMITED (NZ) 2007-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032455-A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents NAPRT, NTPCR, PNP HCAR3 793/4885ALDH1A1 184/4885KDM4E 1572/4885
US-20100010094-A1 Novel nitrophenyl mustard and nitrophenylaziridine alcohols and their corresponding phosphates and their use as targeted cytotoxic agents NAPRT, NTPCR, QDPR HCAR3 589/4885ALDH1A1 164/4885KDM4E 1225/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.