SCHEMBL3591508

SCHEMBL3591508

Nc1[c]ccc([N+](=O)[O-])c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.48
TDP1 Q9NUW8 7/20 0.48
CYP3A4 P08684 4/20 0.47
TSHR P16473 3/20 0.46
LMNA P02545 2/20 0.46
GAA P10253 1/20 0.46
THRB P10828 1/20 0.46
HTT P42858 1/20 0.43
ALOX15 P16050 2/20 0.42
HSD17B10 Q99714 1/20 0.41
MEN1 O00255 2/20 0.40
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
RAB9A P51151 1/20 0.40
TLR9 Q9NR96 1/20 0.40
POLB P06746 1/20 0.39
PTPRC P08575 1/20 0.39
S100A4 P26447 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26325 0.77 TSHR (0.48) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL887743 0.75 TSHR (0.48) ALDH1A1TDP1TSHRLMNAGAA
SCHEMBL1473759 0.75 ALDH1A1 (0.47) ALDH1A1TDP1CYP3A4TSHRLMNA
Water SCHEMBL28995322 0.75 TSHR (0.46) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL57963 0.75 HSD17B10 (0.50) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL455697 0.75 ALDH1A1 (0.50) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL146835 0.75 ALDH1A1 (0.47) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL16005234 0.75 TSHR (0.46) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL10383515 0.75 TSHR (0.46) ALDH1A1TDP1CYP3A4TSHRLMNA
SCHEMBL11425982 0.75 TSHR (0.51) ALDH1A1TDP1CYP3A4TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114213353-A Aryl-oxazole-oxazoline compound and preparation method and application thereof 贵州大学 2022-03-22 CN claimed
CN-103228633-A Heterocyclic compounds as DGAT1 inhibitors PIRAMAL LIFE SCIENCES LTD 2013-07-31 CN claimed
EP-1910320-A2 INTERMEDIATE COMPOUND FOR SYNTHESIZING PHARMACEUTICAL AGENT AND PRODUCTION METHOD THEREOF Mitsubishi Tanabe Pharma Corporation (JP) 2008-04-16 EP claimed
WO-2007011065-A2 INTERMEDIATE COMPOUND FOR SYNTHESIZING PHARMACEUTICAL AGENT AND PRODUCTION METHOD THEREOF MITSUBISHI TANABE PHARMA CORPORATION (JP) 2007-01-25 WO claimed
EP-1289954-B1 SERINE PROTEASE INHIBITORS LILLY CO ELI (US) 2005-09-14 EP claimed
EP-1289953-B1 SERINE PROTEASE INHIBITORS LILLY CO ELI (US) 2005-09-07 EP claimed
US-6936611-B2 Serine protease inhibitors ELI LILLY AND COMPANY (US) 2005-08-30 US claimed
EP-1289972-B1 SERINE PROTEASE INHIBITORS LILLY CO ELI (US) 2004-09-08 EP claimed
EP-1289950-B1 SERINE PROTEASE INHIBITORS LILLY CO ELI (US) 2004-09-08 EP claimed
EP-0031708-B1 CEPHALOSPORIN DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND INTERMEDIATES THEREFOR ICI PHARMA (FR) 1984-06-13 EP claimed
CN-114213353-B Aryl-oxazole-oxazoline compound and preparation method and application thereof 贵州大学 2023-04-14 CN disclosed
CN-115515934-A NAMPT modulators 赛特凯恩蒂克公司 2022-12-23 CN disclosed
CN-114213353-A Aryl-oxazole-oxazoline compound and preparation method and application thereof 贵州大学 2022-03-22 CN disclosed
CN-108610285-B Acetophenone compound, preparation method thereof and application thereof in preventing and treating fatty liver 上海柏翱纳吉医药科技有限公司 2020-04-28 CN disclosed
CN-102245609-B Can be used as the Imidazopyridazine formonitrile HCN of kinase inhibitor BRISTOL-MYERS SQUIBB CO. (US) 2016-03-09 CN disclosed
US-4337061-A NITRO DYES IN AQUEOUS SOLUTION SOCIETE ANONYME DITE: L'OREAL (FR) 1982-06-29 US disclosed
US-4329504-A COUPLERS FOR DYES, HAIR DYES SOCIETE ANONYME DITE: L'OREAL (FR) 1982-05-11 US disclosed
EP-0031708-A2 Cephalosporin derivatives, processes for their manufacture, pharmaceutical compositions containing them and intermediates therefor ICI PHARMA (FR) 1981-07-08 EP disclosed
US-4259261-A OXIDATION COLOR DYES FOR HAIR L'OREAL (FR) 1981-03-31 US disclosed
US-4025642-A ANTIALLERGENS SMITHKLINE CORPORATION (US) 1977-05-24 US disclosed