SCHEMBL359420

SCHEMBL359420

COC(=O)c1cccc2cn(C3CCN(C(=O)OC(C)(C)C)CC3)nc12

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.45
IRAK4 Q9NWZ3 2/20 0.44
EED O75530 1/20 0.43
RBBP4 Q09028 1/20 0.43
SUZ12 Q15022 1/20 0.43
EZH2 Q15910 1/20 0.43
AEBP2 Q6ZN18 1/20 0.43
ALDH1A1 P00352 1/20 0.42
GPR119 Q8TDV5 2/20 0.42
DDB1 Q16531 1/20 0.42
CRBN Q96SW2 1/20 0.42
BACE1 P56817 1/20 0.42
STS P08842 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN6 P29350 1/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29267085 0.81 PARP1 (0.39) PARP1EEDRBBP4SUZ12EZH2
SCHEMBL28614035 0.81 PARP1 (0.52) PARP1ALDH1A1GPR119
SCHEMBL358681 0.80 EED (0.46) PARP1EEDRBBP4SUZ12EZH2
SCHEMBL20135591 0.79 GPR119 (0.50) IRAK4GPR119DDB1CRBNPTPN2
SCHEMBL2270749 0.79 CCNT1 (0.41) PARP1EEDRBBP4SUZ12EZH2
SCHEMBL20606506 0.78 IRAK4 (0.46) IRAK4EEDRBBP4SUZ12EZH2
SCHEMBL358920 0.78 NR3C1 (0.43) PARP1EEDRBBP4SUZ12EZH2
SCHEMBL25104075 0.78 NR1H2 (0.41) IRAK4EEDRBBP4SUZ12EZH2
SCHEMBL30158059 0.78 MAPT (0.44) IRAK4ALDH1A1GPR119DDB1CRBN
SCHEMBL28624126 0.77 PARP1 (0.55) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012006958-A1 AMIDS SUBSTITUTED INDAZOLE DERIVATIVEES AS PLOY(ADP-RIBOSE)POLYMERASE INHIBITORS ZHEJIANG BETA PHARMA INC. (CN) 2012-01-19 WO disclosed