SCHEMBL3595140

SCHEMBL3595140

CCOC(=O)Cc1cccnc1C

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.48
TBXAS1 P24557 1/20 0.48
LMNA P02545 2/20 0.48
PKM P14618 1/20 0.47
MAPK1 P28482 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TP53 P04637 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
FFAR1 O14842 1/20 0.45
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
P2RX7 Q99572 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
BRD4 O60885 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20037256 0.86 PAM (0.50) MAPTTBXAS1LMNAMAPK1KDM4E
SCHEMBL14678422 0.85 P2RX7 (0.47) MAPTLMNAPKMALDH1A1KDM4E
SCHEMBL9370451 0.84 MAPT (0.49) MAPTTBXAS1LMNAPKMMAPK1
SCHEMBL4061267 0.84 MAPT (0.52) MAPTTBXAS1LMNAPKMMAPK1
SCHEMBL27563569 0.84 SMN1; SMN2 (0.47) MAPTTBXAS1LMNAPKMMAPK1
SCHEMBL8664219 0.84 CYP4F2 (0.60) MAPTLMNAALDH1A1KDM4EHSD17B10
SCHEMBL3587106 0.84 MAPT (0.46) MAPTTBXAS1LMNAPKMMAPK1
SCHEMBL6642153 0.84 MAPT (0.46) MAPTTBXAS1LMNAPKMMAPK1
SCHEMBL30178346 0.84 CYP4F2 (0.60) MAPTLMNAALDH1A1KDM4EHSD17B10
SCHEMBL24767639 0.83 P2RX7 (0.46) MAPTLMNAALDH1A1KDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109716491-B Method for manufacturing field effect transistor and method for manufacturing wireless communication device 东丽株式会社 2023-06-09 CN disclosed
CN-110156672-B Preparation method of semicarbazide compound and application of prepared compound 浙江师范大学 2022-06-10 CN disclosed
CN-110156672-B Preparation method of semicarbazide compound and application of prepared compound 浙江师范大学 2022-06-10 CN disclosed
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
WO-2018065607-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2018-04-12 WO disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed
EP-3305781-A1 CHEMICAL SUBSTANCES WHICH INHIBIT THE ENZYMATIC ACTIVITY OF HUMAN KALLIKREIN-RELATED PEPTIDASE 6 (KLK6) Deutsches Krebsforschungszentrum (DE) 2018-04-11 EP disclosed
US-9085572-B2 4-(pyridin-3-yl)-2(pyridin-2yl)-1,2-dihydro-3H-pyrazol-3-one derivatives as specific HIF-pyrolyl-4-hydroxylase inhibitors for treating cardiovascular and haematological diseases BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-21 US disclosed
US-9085572-B2 4-(pyridin-3-yl)-2(pyridin-2yl)-1,2-dihydro-3H-pyrazol-3-one derivatives as specific HIF-pyrolyl-4-hydroxylase inhibitors for treating cardiovascular and haematological diseases BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-21 US disclosed
US-9085572-B2 4-(pyridin-3-yl)-2(pyridin-2yl)-1,2-dihydro-3H-pyrazol-3-one derivatives as specific HIF-pyrolyl-4-hydroxylase inhibitors for treating cardiovascular and haematological diseases BAYER INTELLECTUAL PROPERTY GMBH (DE) 2015-07-21 US disclosed
US-6242458-B1 INHIBITING FARNESYL PROTEIN TRANSFERASE IN A HUMAN SCHERING CORPORATION 2001-06-05 US disclosed
US-5891872-A INHIBIT FARNESYL-PROTEIN TRANSFERASE SCHERING CORPORATION (US) 1999-04-06 US disclosed
US-5807852-A Tricyclic amide and urea compounds useful for inhibition of G-protein function and for treatment of proliferative diseases SCHERING CORPORATION (US) 1998-09-15 US disclosed
US-5807853-A Tricyclic amide and urea compounds, useful inhibition of g-protein function and for treatment of proliferative diseases SCHERING CORPORATION (US) 1998-09-15 US disclosed
US-5719148-A FARNESYL-PROTEIN TRANSFERASE INHIBITORS SCHERING CORPORATION (US) 1998-02-17 US disclosed
US-5714609-A FORMING CHEMICAL INTERMEDIATE BY NITRATING SUBSTITUTED BENZO/5,6/CYCLOHEPTA/1,2-B/PYRIDINE WITH TETRABUTYLAMMONIUM NITRATE AND TRIFLUOROACETIC ANHYDRIDE IN SOLVENT AT REDUCED TEMPERATURE SCHERING CORPORATION (US) 1998-02-03 US disclosed
US-5700806-A FARNESYL PROTEIN TRANSFERASE ENZYME INHIBITOR, ANTITUMOR AGENTS SCHERING CORPORATION (US) 1997-12-23 US disclosed
US-5696121-A 4-(3-BROMO 8-CHLORO-6,11-DIHYDRO-5H-BENZO(5,6)CYCLOHEPTA(1,2B)PYRIDINE-11-YL)-N-(3 -PYRIDINYL)-1-PIPERAZINECARBOXIDE; ANTITUMOR AGENT; FARNESYL PROTEIN TRANSFERASE INHIBITOR SCHERING CORPORATION (US) 1997-12-09 US disclosed
EP-0723540-A1 TRICYCLIC AMIDE AND UREA COMPOUNDS USEFUL FOR INHIBITION OF G-PROTEIN FUNCTION AND FOR TREATMENT OF PROLIFERATIVE DISEASES SCHERING CORPORATION (US) 1996-07-31 EP disclosed
WO-1995010516-A1 TRICYCLIC AMIDE AND UREA COMPOUNDS USEFUL FOR INHIBITION OF G-PROTEIN FUNCTION AND FOR TREATMENT OF PROLIFERATIVE DISEASES SCHERING CORPORATION (US) 1995-04-20 WO disclosed