SCHEMBL3595249

SCHEMBL3595249

NCc1c(-c2ccc(Cl)cc2Cl)ncn1Cc1ccc(-c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 8/20 0.47
CYP3A4 P08684 2/20 0.46
MDM4 O15151 2/20 0.46
TP53 P04637 2/20 0.46
MDM2 Q00987 2/20 0.46
CSNK2A1 P68400 2/20 0.44
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
TAAR1 Q96RJ0 1/20 0.43
GRM2 Q14416 1/20 0.41
DPP8 Q6V1X1 2/20 0.41
CYP2C19 P33261 1/20 0.40
DPP9 Q86TI2 1/20 0.40
NSD2 O96028 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3079559 0.93 DPP4 (0.51) DPP4CYP3A4MDM4TP53MDM2
SCHEMBL3091375 0.90 DPP4 (0.47) DPP4CYP3A4MDM4TP53MDM2
SCHEMBL3096840 0.86 DPP4 (0.46) DPP4CYP3A4MDM4TP53MDM2
SCHEMBL3595741 0.86 DPP4 (0.44) DPP4CYP3A4MDM4TP53MDM2
SCHEMBL3091436 0.86 DPP4 (0.46) DPP4CYP3A4CYP11B1CYP11B2DPP8
SCHEMBL3102277 0.86 DPP4 (0.44) DPP4MDM4TP53MDM2DPP8
SCHEMBL3606001 0.84 DPP4 (0.44) DPP4CYP3A4DPP8DPP9
SCHEMBL3089796 0.84 DPP4 (0.44) DPP4MDM4MDM2DPP8
SCHEMBL3084580 0.83 DPP4 (0.49) DPP4CYP3A4DPP8
SCHEMBL3595932 0.83 DPP4 (0.49) DPP4CYP3A4TP53DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed