SCHEMBL3595401

SCHEMBL3595401

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CCc1c[nH]c2cc(F)ccc12

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.46
HTR1A P08908 1/20 0.40
GPR84 Q9NQS5 2/20 0.39
CDK4 P11802 3/20 0.38
CCND1 P24385 3/20 0.38
MDM2 Q00987 3/20 0.37
MDM4 O15151 2/20 0.37
TP53 P04637 2/20 0.37
SSTR4 P31391 3/20 0.37
SSTR2 P30874 2/20 0.37
DPP4 P27487 2/20 0.36
DPP8 Q6V1X1 1/20 0.36
TRPM8 Q7Z2W7 2/20 0.36
MPO P05164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3088301 0.89 HTR2A (0.46) HTR2AGPR84CDK4CCND1MDM2
SCHEMBL3604686 0.88 DPP4 (0.41) HTR2AGPR84CDK4CCND1TP53
SCHEMBL3598443 0.85 HTR2A (0.42) HTR2AHTR1AGPR84CDK4CCND1
SCHEMBL3596995 0.85 SLC6A4 (0.41) HTR2AGPR84CDK4CCND1MDM2
SCHEMBL3606760 0.80 DPP4 (0.44) TP53DPP4DPP8
SCHEMBL3096850 0.80 DPP4 (0.44) DPP4DPP8
SCHEMBL3604409 0.78 DPP4 (0.45) DPP4DPP8
SCHEMBL3607898 0.78 MDM2 (0.46) HTR2AGPR84CDK4CCND1MDM2
SCHEMBL3092513 0.77 DPP4 (0.47) DPP4DPP8
SCHEMBL3084453 0.76 CNR1 (0.45) DPP4DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed