SCHEMBL3604686

SCHEMBL3604686

NCc1c(-c2ccc(Cl)cc2Cl)ncn1CCc1c[nH]c2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.41
GOT1 P17174 1/20 0.41
HTR2A P28223 3/20 0.41
MPO P05164 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
NFKB1 P19838 1/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41
HTR2C P28335 1/20 0.41
HTR7 P34969 1/20 0.41
CTSK P43235 1/20 0.41
HTR6 P50406 1/20 0.41
CYP2A13 Q16696 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
CDK4 P11802 2/20 0.41
CCND1 P24385 2/20 0.41
TRPM8 Q7Z2W7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3595401 0.88 HTR2A (0.46) DPP4HTR2AMPOCDK4CCND1
SCHEMBL3088301 0.88 HTR2A (0.46) DPP4HTR2AHTR1DCDK4CCND1
SCHEMBL3605880 0.85 MDM4 (0.43) GOT1HTR2AHTR1DHTR1BHTR2C
SCHEMBL3596995 0.83 SLC6A4 (0.41) DPP4HTR2AHTR2CCDK4CCND1
SCHEMBL3092513 0.83 DPP4 (0.47) DPP4CYP3A4TAAR1
SCHEMBL3096850 0.82 DPP4 (0.44) DPP4CYP3A4
SCHEMBL3604409 0.81 DPP4 (0.45) DPP4CYP3A4TAAR1
SCHEMBL3604955 0.80 DPP4 (0.48) DPP4CYP1A2CYP3A4CYP2D6NPC1
SCHEMBL3600802 0.78 DPP4 (0.44) DPP4
SCHEMBL3595072 0.77 DPP4 (0.46) DPP4CYP1A2CYP3A4CYP2D6RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7728146-B2 Enzyme inhibitors PROBIODRUG AG (DE) 2010-06-01 US claimed